Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
All Genders
NCT07417189

A Phase I/II Study of ABSK141 in Patients With Advanced Solid Tumors ( ABSK141-101 )

Led by Abbisko Therapeutics Co, Ltd · Updated on 2026-03-11

401

Participants Needed

1

Research Sites

178 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

This is a first-in-human (FIH), exploratory, multicenter, open-label, phase I/II study of ABSK141 in patients with advanced solid tumors to to evaluate safety, tolerability, PK and optimize the dosage.

CONDITIONS

Official Title

A Phase I/II Study of ABSK141 in Patients With Advanced Solid Tumors ( ABSK141-101 )

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Patients must understand and sign informed consent before screening
  • Male or female age 18 years or older
  • Histologically confirmed locally advanced or metastatic solid tumors
  • For escalation backfill cohorts: solid tumors with KRAS G12D mutation including colorectal cancer, non-small cell lung cancer, or pancreatic ductal adenocarcinoma
  • Must have at least one measurable target lesion according to RECIST 1.1
  • For expansion part: solid tumors with KRAS G12D mutation including colorectal cancer, non-small cell lung cancer, pancreatic ductal adenocarcinoma, or other solid tumors
  • For phase II: locally advanced or metastatic solid tumors with disease progression after or intolerance to standard treatment, or no standard treatment available
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
  • Adequate organ and bone marrow function per screening within 14 days before first dose
  • For food effect exploration participants: able to eat a standardized high-fat, high-calorie meal within 30 minutes and fast for 10 hours
Not Eligible

You will not qualify if you...

  • Known allergy or hypersensitivity to any component of ABSK141
  • Previous treatment with investigational KRAS G12D inhibitors, pan- or multi-RAS inhibitors, or direct RAS-targeted therapy (for backfill cohorts and expansion part)
  • Active additional progressing malignancy requiring treatment
  • Unable to swallow capsules or tablets or have significant gastrointestinal disorders affecting absorption
  • Anti-tumor therapy within 2 weeks or 5 half-lives (whichever is shorter), or radiotherapy/antibody therapy within 4 weeks before study
  • Major surgery within 4 weeks before first dose with unhealed wounds or infections
  • Prior toxicities from cancer therapies not resolved to Grade 1 or less
  • Use of proton pump inhibitors or certain CYP3A and P-gp inhibitors/inducers within specified timeframes
  • Active central nervous system metastases
  • History of interstitial lung disease requiring steroids
  • Significant cardiac disease
  • Non-small cell lung cancer patients with other driver mutations without targeted therapy
  • Known HIV infection or AIDS-related illness
  • Hepatitis infection
  • Uncontrolled ascites or pleural effusion
  • Pregnant or nursing women
  • Refusal to use effective birth control during and after study
  • Vaccination with live attenuated vaccines within 4 weeks before first dose
  • Planned major surgery during study
  • Any other clinically significant comorbidities

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

1
2
3
+1

Trial Site Locations

Total: 1 location

1

Fudan University Shanghai Cancer Center

Shanghai, China, 201321

Actively Recruiting

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Research Team

Y

Yu Zhang, Bachelor

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

6

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