Actively Recruiting

Phase 2
Age: 18Years +
MALE
ID07005154

A Phase 2 Open-label Multi-cohort Study to Assess the Safety and Efficacy of ASP5541 in Men With Advanced Prostate Cancer

Led by Astellas Pharma Global Development, Inc. · Updated on 2026-05-01

218

Participants Needed

33

Research Sites

N/A

Total Duration

On this page

AI-Summary

What this Trial Is About

Researchers are evaluating the safety and effectiveness of ASP5541, a new injectable form of abiraterone acetate, in men with advanced prostate cancer. This study focuses on men with metastatic hormone-sensitive prostate cancer (mHSPC) or metastatic castration-resistant prostate cancer (mCRPC) who have not previously been treated with androgen receptor pathway inhibitors (ARPIs). The study aims to compare ASP5541 with the standard oral abiraterone acetate combined with prednisone or prednisolone and assess ASP5541's safety alone and with steroids. Participants are divided into three groups: men with mCRPC receiving either ASP5541 plus prednisone/prednisolone or abiraterone acetate plus prednisone/prednisolone; men with mHSPC receiving either ASP5541 alone or abiraterone acetate plus prednisone/prednisolone; and Japanese men with mCRPC or mHSPC receiving ASP5541 with prednisone/prednisolone. ASP5541 is given by intramuscular injection every 12 weeks, prednisone/prednisolone is taken orally once or twice daily depending on cancer type, and abiraterone acetate is taken daily as a tablet. All participants continue standard care, including androgen deprivation therapy. During and after treatment, participants will have regular clinic visits for health checks, scans to monitor cancer progression, and safety assessments. Some men will monitor blood pressure weekly at home. Researchers will measure outcomes such as prostate-specific antigen (PSA) levels, adverse events, heart function, and overall health status up to several years. The study includes long-term follow-up to assess progression-free survival and treatment responses.

CONDITIONS

Brief Title

A Phase 2 Study to Evaluate the Effects of ASP5541 in Participants With Prostate Cancer

Who Can Participate

Age: 18Years +
MALE

Eligibility Criteria

Eligible

You may qualify if you...

  • Male participant diagnosed with adenocarcinoma of the prostate without neuroendocrine or small cell features
  • ECOG performance status 0 or 1, or 2 if due to bone pain
  • Estimated life expectancy of at least 12 months for mHSPC or 6 months for mCRPC
  • Able to understand and follow all study procedures
  • Diagnosed with metastatic castration-resistant or hormone-sensitive prostate cancer confirmed by imaging
  • Currently receiving androgen deprivation therapy or has had surgical castration; mHSPC participants must have started castration therapy at least 14 days before first treatment
  • For mCRPC, evidence of disease progression by imaging or rising PSA levels
  • For mCRPC, serum testosterone level below 1.73 nmol/L at screening
  • Male participants agree to use contraception or abstain during treatment and for 7 months after final dose
  • Male participants agree not to donate sperm during treatment and for 7 months after final dose
  • Not participating in another interventional study during this trial
  • Normal serum potassium at screening without supplementation
Not Eligible

You will not qualify if you...

  • Any disease, infection, or condition that increases risk or complicates study participation
  • Active central nervous system metastases unless treated and stable
  • Other active cancers requiring treatment, except certain treated skin or early-stage cancers in remission
  • Significant heart conditions including poorly controlled arrhythmias, long QT syndrome, recent heart attack, or heart failure greater than NYHA Class II
  • Uncontrolled hypertension as defined by specific blood pressure thresholds
  • Recent arterial or venous thrombotic or embolic events within specified timeframes
  • Ongoing Grade > 2 adverse events or unresolved toxicities
  • Recent major surgery or planned surgery during study participation
  • Recent febrile illness or active infection within 28 days before treatment
  • Recent blood transfusion within 1 month before treatment
  • Impaired pituitary or adrenal function
  • High hemoglobin A1c levels indicating uncontrolled diabetes
  • Current active liver disease or moderate to severe hepatic impairment
  • Known HIV infection
  • Body mass index over 40 kg/m2
  • Drug or alcohol abuse within 2 years before screening
  • Recent use of systemic glucocorticoids over 10 mg prednisone equivalent
  • Recent use of herbal medications affecting prostate or cancer
  • Current treatment with certain hormone therapies or CYP inhibitors
  • Use of prohibited medications
  • Specific prior treatments within defined timeframes before enrollment
  • Prior treatment with ASP5541
  • Low blood counts or abnormal laboratory values
  • Known hypersensitivity to study drugs
  • Gastrointestinal disorders affecting drug absorption or metabolism
  • For mCRPC and mHSPC, treatment history restrictions as specified in protocol details
  • Participation in another investigational therapy within 4 weeks before study start

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person)

Treatment

Duration - Up to 37 months

Participants receive active drug treatments including ASP5541 every 12 weeks, prednisone or prednisolone orally twice daily, abiraterone acetate orally once daily, or a combination depending on cohort assignment.

Visits every 12 weeks aligned with ASP5541 dosing and additional visits for oral medication monitoring

Follow-up

Duration - Up to 84 months

Participants are monitored for safety, adverse events, and treatment efficacy after treatment completion.

Periodic visits for up to 84 months

Trial Site Locations

Total: 33 locations

1

Clearview Cancer Institute

Huntsville, Alabama, United States, 35805

Actively Recruiting

2

H. Lee Moffitt Cancer Center

Tampa, Florida, United States, 33612

Actively Recruiting

3

Associated Urological Specialists

Chicago Ridge, Illinois, United States, 60415

Actively Recruiting

4

Ochsner Health - Ochsner Medical Center - New Orleans

New Orleans, Louisiana, United States, 70121

Actively Recruiting

5

New Mexico Oncology Hematology Consultants

Albuquerque, New Mexico, United States, 87109

Actively Recruiting

6

Solaris Health - The Urology Group

Cincinnati, Ohio, United States, 45212

Actively Recruiting

7

Carolina Urologic Research Center

Myrtle Beach, South Carolina, United States, 29572

Actively Recruiting

8

Tennessee Oncology Nashville

Nashville, Tennessee, United States, 37203

Actively Recruiting

9

University of Virginia Cancer Center

Charlottesville, Virginia, United States, 22908-07

Actively Recruiting

10

UW Health Carbone Cancer Center

Madison, Wisconsin, United States, 53792

Actively Recruiting

11

Subei People's Hospital

Yangzhou, Jiangsu, China, 225001

Actively Recruiting

12

The Second Hospital of Tianjin Medical University

Tianjin, Tianjin Municipality, China, 300211

Actively Recruiting

13

Huai'an First People's Hospital

Huaian, China, 211731

Actively Recruiting

14

Renji Hospital Shanghai Jiaotong Univ School of Medicine

Shanghai, China, 200127

Actively Recruiting

15

Site FR33004

Strasbourg, France

Actively Recruiting

16

Site DE49004

Nürtingen, Baden-Wurttemberg, Germany

Actively Recruiting

17

Site DE49001

Heinsberg, Germany

Actively Recruiting

18

National Cancer Center Hospital East

Kashiwa, Chiba, Japan

Actively Recruiting

19

Shizuoka Cancer Center

Sunto-gun, Shizuoka, Japan

Actively Recruiting

20

Nippon Medical School Hospital

Bunkyo-ku, Tokyo, Japan

Actively Recruiting

21

The Cancer Institute Hospital of JFCR

Koto, Tokyo, Japan

Actively Recruiting

22

Harasanshin Hospital

Fukuoka, Japan

Actively Recruiting

23

Osaka International Cancer Institute

Osaka, Japan

Actively Recruiting

24

PanOncology Trials

San Juan, Puerto Rico

Actively Recruiting

25

Site KR82008

Gwangju, South Korea

Actively Recruiting

26

Site KR82002

Seoul, South Korea

Actively Recruiting

27

Site KR82003

Seoul, South Korea

Actively Recruiting

28

Site KR82004

Seoul, South Korea

Actively Recruiting

29

Site KR82007

Seoul, South Korea

Actively Recruiting

30

Site ES34006

Barcelona, Catalonia, Spain

Actively Recruiting

31

Site TW88603

Kaohsiung City, Taiwan

Actively Recruiting

32

Site TW88602

Taipei, Taiwan

Actively Recruiting

33

Site GB44003

London, United Kingdom

Actively Recruiting

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Research Team

A

Astellas Pharma Global Development, Inc.

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

6

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