Actively Recruiting

Phase 1
Age: 20Years +
All Genders
NCT04608110

A Phase 1 Trial of ASTX030 in Patients With Myelodysplastic Syndrome

Led by Taiho Pharmaceutical Co., Ltd. · Updated on 2025-12-03

40

Participants Needed

10

Research Sites

269 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

The purpose of this study is to identify the doses of the oral azacitidine formulations and cedazuridine (CED) tablets which achieve a total AUC for AZA comparable to that for AZA injection at 75 mg/m2

CONDITIONS

Official Title

A Phase 1 Trial of ASTX030 in Patients With Myelodysplastic Syndrome

Who Can Participate

Age: 20Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Patients aged 20 years or older
  • Diagnosis of Myelodysplastic Syndrome (MDS) including RA, RARS, RAEB, RAEB-T, or CMML by FAB classification
  • Low or intermediate-1 risk patients by IPSS only if unlikely to respond to other treatment or currently treated with azacitidine injection
  • ECOG performance status score of 0 or 1, or 2 due to primary disease
  • Adequate hepatic function: total bilirubin ≤ 2.0 × ULN; AST ≤ 2.5 × ULN; ALT ≤ 2.5 × ULN
  • Adequate renal function: serum creatinine ≤ 1.5 × ULN or creatinine clearance/glomerular filtration rate ≥ 50 mL/min
  • Respiratory function with oxygen saturation (SpO2) ≥ 90%
  • Expected survival of at least 3 months
  • Provided written informed consent
Not Eligible

You will not qualify if you...

  • Unlikely to respond to azacitidine
  • Received chemotherapy, hormone therapy, antibody therapy, radiotherapy, or other anticancer treatments within 3 weeks before first study drug dose
  • Used any other investigational medicinal product or privately imported medicine within 4 weeks before first study drug dose
  • Heart disease classified as New York Heart Association Class 3 or 4
  • Uncontrolled systemic disease or active infection
  • Uncontrolled gastric or duodenal ulcer
  • Prior or current interstitial lung disease
  • History of surgical gastrectomy
  • Life-threatening conditions, multiple organ failure, or factors affecting safety or drug metabolism
  • Other malignancies except certain treated or stable cancers
  • Positive for HIV antibody, HBV-DNA, or HCV antibody
  • Grade 2 or higher adverse events from prior treatment (except alopecia)
  • Recent highly invasive surgery within 4 weeks before first study drug dose
  • Previous or planned hematopoietic stem cell transplantation
  • History of hypersensitivity to study drug or its components
  • High risk for protocol noncompliance due to mental disorders or substance abuse
  • Pregnant or nursing females, or positive pregnancy test at screening
  • Sexually active males or females of childbearing potential not agreeing to use two birth control methods or abstinence during and after trial
  • Investigator judgment deeming patient otherwise ineligible

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 10 locations

1

Nippon Medical School Hospital

Bunkyō City, Japan

Actively Recruiting

2

Fukushima Medical University Hospital

Fukushima, Japan

Actively Recruiting

3

Saitama Medical University Hospital

Iruma, Japan

Actively Recruiting

4

University Hospital, Kyoto Prefectural University of Medicine

Kyoto, Japan

Actively Recruiting

5

Nagasaki University Hospital

Nagasaki, Japan

Actively Recruiting

6

Osaka City General Hospital

Osaka, Japan

Actively Recruiting

7

Kindai University Hospital

Sakai, Japan

Actively Recruiting

8

NTT Medical Center Tokyo

Shinagawa-Ku, Japan

Actively Recruiting

9

Tokyo Medical University Hospital

Shinjuku-Ku, Japan

Actively Recruiting

10

Yamagata University Hospital

Yamagata, Japan

Actively Recruiting

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Research Team

D

Drug Information Center

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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