Actively Recruiting

Phase 1
Age: 18Years +
MALE
NCT04729114

A Safety and Dose-finding Study of PRL-02 Depot in Men With Advanced Prostate Cancer

Led by Astellas Pharma Global Development, Inc. · Updated on 2026-02-04

174

Participants Needed

25

Research Sites

415 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

Medicines that reduce the amount of testosterone in the body are commonly used to treat prostate cancer. PRL-02 depot is a potential treatment for men with advanced prostate cancer. It is given by an injection into the muscle. Men with advanced prostate cancer can take part in this study. Their cancer has come back after previous cancer treatment, or the previous cancer treatment they had didn't work. The main aims of the study are: * to check the safety of PRL-02 depot given with and without another medicine called enzalutamide. * to check if the men can tolerate PRL-02 depot given with or without enzalutamide. * to find a suitable dose of PRL-02 depot. This study will be in 2 parts. In the first part, different small groups of men will receive lower to higher doses of PRL-02 depot together with other medicines. In the second part of the study, men who have previously taken a hormone therapy called abiraterone acetate or have previously taken 1 specific hormone therapy as part of their prostate cancer treatment can take part. Men in both parts of the study will receive injections of PRL-02 depot into a muscle once every 12 weeks. They will also take dexamethasone or prednisone, or enzalutamide once a day. The other medicines they take depend on which group and which part of the study they are in. During the study, the men will visit the clinic several times for health checks and scans. After the final visit, men whose cancer has not become worse will continue to have health checks and scans every few months.

CONDITIONS

Official Title

A Safety and Dose-finding Study of PRL-02 Depot in Men With Advanced Prostate Cancer

Who Can Participate

Age: 18Years +
MALE

Eligibility Criteria

Eligible

You may qualify if you...

  • Histological evidence of adenocarcinoma of the prostate
  • For dose escalation groups, documented metastatic castration-sensitive or castration-resistant prostate cancer
  • Evidence of disease progression by scans or PSA levels as defined
  • Prior hormone therapy requirements depend on study group
  • Serum testosterone level below 50 ng/dL for mCRPC participants
  • Adequate muscle mass for injection and ECOG performance status of 0 or 1
  • Adequate bone marrow, kidney, and liver function as specified
  • Serum albumin at least 3 gm/dL and serum potassium at least 3.5 mEq/L
  • Willingness to use effective contraception if sexually active with a female partner of childbearing potential
  • Ability to comply with study requirements throughout the study
  • For Group H, ability to swallow enzalutamide capsules whole
Not Eligible

You will not qualify if you...

  • Known active central nervous system metastases, unless treated and stable
  • Impending bone fracture due to bone metastases
  • Other active malignancies requiring treatment, except certain treated skin or early-stage cancers in remission
  • Significant cardiac diseases including uncontrolled arrhythmias or heart failure above NYHA Class II
  • Uncontrolled hypertension or recent thrombotic events
  • Recent investigational drug or chemotherapy use within specified timeframes
  • Unresolved significant toxicity from prior cancer therapy
  • Recent major surgery or trauma or recent blood transfusion
  • History of pituitary or adrenal gland disorders
  • Prior treatments with abiraterone acetate or certain hormone therapies depending on group
  • Current use of systemic ketoconazole or CYP17 inhibitors, or recent systemic azole drugs
  • Use of estrogens within 12 weeks before study drug
  • Need for systemic glucocorticoids beyond replacement doses
  • Use of herbal products lowering PSA or high-dose biotin supplements
  • Use of strong CYP3A4 inducers except enzalutamide in Group H
  • Known hypersensitivity to study drugs or excipients
  • Active liver disease or infections including hepatitis or uncontrolled HIV
  • Poorly controlled diabetes with high HbA1c
  • Body mass index over 40 kg/m2
  • For Group H, additional cardiac conditions, seizure history, prohibited medication use, gastrointestinal absorption disorders, or hypersensitivity to capsule components

AI-Screening

AI-Powered Screening

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Trial Site Locations

Total: 25 locations

1

Arizona Urology Specialists

Tucson, Arizona, United States, 85715

Withdrawn

2

Los Angeles Cancer Network

Anaheim, California, United States, 92801

Actively Recruiting

3

Providence Medical Group Oncology Santa Rosa

Santa Rosa, California, United States, 95403

Actively Recruiting

4

Florida Urology Partners

Tampa, Florida, United States, 33609

Withdrawn

5

Fort Wayne Medical Oncology and Hematology, Inc.

Fort Wayne, Indiana, United States, 46804

Withdrawn

6

First Urology

Jeffersonville, Indiana, United States, 47130

Actively Recruiting

7

Wichita Urology Group

Wichita, Kansas, United States, 67226

Actively Recruiting

8

National Cancer Institute

Bethesda, Maryland, United States, 20892

Withdrawn

9

Chesapeake Urology

Towson, Maryland, United States, 21204

Actively Recruiting

10

XCancer Center Omaha/Urology Cancer Center

Omaha, Nebraska, United States, 68130

Completed

11

Garden Sate Urology

Morristown, New Jersey, United States, 07960

Withdrawn

12

New Mexico Oncology Hematology Consultants Ltd

Albuquerque, New Mexico, United States, 87109

Actively Recruiting

13

Duke Cancer Center

Durham, North Carolina, United States, 27710

Actively Recruiting

14

Helios Clinical Research, LLC

Middleburg Heights, Ohio, United States, 44130

Withdrawn

15

Toledo Clinical Cancer Center

Toledo, Ohio, United States, 43623

Withdrawn

16

MidLantic Urology

Bala-Cynwyd, Pennsylvania, United States, 19004

Actively Recruiting

17

Carolina Urologic Research Center

Myrtle Beach, South Carolina, United States, 29572

Actively Recruiting

18

Urology Associates PC

Nashville, Tennessee, United States, 37209

Actively Recruiting

19

Urology Clinics of North Texas

Dallas, Texas, United States, 75231

Actively Recruiting

20

Houston Metro Urology

Houston, Texas, United States, 77027

Actively Recruiting

21

Oncology Consultants

Houston, Texas, United States, 77030

Withdrawn

22

Urology San Antonio

San Antonio, Texas, United States, 78229

Withdrawn

23

University of Virginia Cancer Center

Charlottesville, Virginia, United States, 22908

Actively Recruiting

24

Northwest Medical Specialties

Tacoma, Washington, United States, 98405

Actively Recruiting

25

Pan American Center for Oncology Trials, LLC

San Juan, Rio Piedras, Puerto Rico, 00935

Actively Recruiting

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Research Team

A

Astellas Pharma Global Development, Inc.

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

5

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A Safety and Dose-finding Study of PRL-02 Depot in Men With Advanced Prostate Cancer | DecenTrialz