Actively Recruiting

Phase 1
Phase 2
Age: 18Years - 80Years
All Genders
Healthy Volunteers
NCT05395624

Safety, PK and Biodistribution of 18F-OP-801 in Patients With ALS, AD, MS, PD and Healthy Volunteers

Led by Ashvattha Therapeutics, Inc. · Updated on 2025-05-02

65

Participants Needed

3

Research Sites

169 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

This is a Phase 1/2 study to evaluate the safety and tolerability of 18F-OP-801 in subjects with ALS, AD, MS, PD and age-matched HVs. 18F-OP-801 is intended as a biomarker for PET imaging of activated microglia and macrophages in regions of neuroinflammation.

CONDITIONS

Official Title

Safety, PK and Biodistribution of 18F-OP-801 in Patients With ALS, AD, MS, PD and Healthy Volunteers

Who Can Participate

Age: 18Years - 80Years
All Genders
Healthy Volunteers

Eligibility Criteria

Eligible

You may qualify if you...

  • Ability to understand and sign informed consent and privacy forms
  • Female participants of non-childbearing potential must be surgically sterile or postmenopausal
  • Females of childbearing potential and all males must agree to use medically accepted contraception or abstinence during study and follow-up
  • Male subjects must abstain from sperm donation during study and 90 days after Day 1
  • Female subjects may not be pregnant, lactating, or breastfeeding
  • Female subjects of childbearing potential must have negative pregnancy tests at screening and check-in
  • Estimated glomerular filtration rate (eGFR) above 45 mL/min/1.73m2 at screening
  • C-reactive protein level at or below 10 mg/dL
  • Willingness and ability to comply with all study requirements
  • ALS subjects aged 18 to 80 with diagnosed ALS according to modified El Escorial criteria
  • ALS subjects must have forced vital capacity of 50% or greater or be able to lie flat for up to 90 minutes
  • AD subjects aged 40 to 80 with clinical diagnosis of early stage Alzheimer's dementia and positive biomarkers
  • AD subjects must have MMSE score above 20 at screening
  • MS subjects aged 18 to 70 with diagnosis and medication changes discussed with Medical Monitor
  • RRMS subjects must meet 2017 McDonald criteria and have documented relapse or MRI lesions as specified
  • Progressive MS subjects must meet 2017 McDonald criteria with disability scores and no relapse in prior 6 months
  • PD subjects aged 55 to 80 with diagnosis of definite idiopathic Parkinson's disease
  • PD medication changes discussed with Medical Monitor
Not Eligible

You will not qualify if you...

  • Body weight over 120 kg
  • Significant past or current medical conditions affecting drug metabolism or safety as judged by investigator
  • History of recurrent kidney or liver cancer
  • Pacemaker, defibrillator, or incompatible metallic implants
  • Inability to lie still in PET/CT or PET/MRI scanner for up to 90 minutes
  • Clinically significant abnormal laboratory results at screening or check-in
  • Recent acute illness within 10 days before screening
  • History of alcoholism or drug abuse within 2 years prior to screening
  • Positive drug or cotinine tests at screening or check-in
  • Recent immunizations within 28 days prior to screening
  • Use of other investigational drugs within 30 days or 5 half-lives before Day 1
  • Corticosteroid treatment within 30 days before baseline
  • Use of certain NSAIDs within 14 days before Day 1
  • Significant blood loss or donation within 30 days before screening
  • MRI or CT findings that interfere with imaging interpretation
  • Investigator judgment of inability to meet study schedule or safety concerns
  • MS-specific exclusions including neuromyelitis optica, MOG encephalomyelitis, or PML
  • PD-specific exclusions including secondary, atypical, or genetic parkinsonism
  • Healthy volunteer exclusions including relevant neurological findings, family history, or CNS disorders

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 3 locations

1

UCSF

San Francisco, California, United States, 94107

Actively Recruiting

2

Stanford University

Stanford, California, United States, 94305

Actively Recruiting

3

Mayo Clinic Jacksonville

Jacksonville, Florida, United States, 32224

Actively Recruiting

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Research Team

J

Julee Cheung

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

PARALLEL

Primary Purpose

DIAGNOSTIC

Number of Arms

5

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