Actively Recruiting

Phase 1
Age: 18Years - 55Years
All Genders
Healthy Volunteers
NCT06082323

A Single and Multiple Ascending Dose Trial of LT-002-158 Tablets in Healthy Adult Volunteers

Led by Leadingtac Pharmaceutical (Shaoxing) Co., Ltd. · Updated on 2025-02-19

127

Participants Needed

1

Research Sites

50 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

LT-002-158 is an oral IRAK4 protein degrader being developed for the treatment of autoimmune disease and inflammation including Hidradenitis Suppurativa and Atopic Dermatitis. This first-in-human (FIH) study will characterize the safety, tolerability and the pharmacokinetics/pharmacodynamics (PK/PD) of a single ascending dose and multiple ascending doses of LT-002-158 in healthy volunteers. The effects of food on the pharmacokinetics of LT-002-158 will also be assessed in healthy volunteers.

CONDITIONS

Official Title

A Single and Multiple Ascending Dose Trial of LT-002-158 Tablets in Healthy Adult Volunteers

Who Can Participate

Age: 18Years - 55Years
All Genders
Healthy Volunteers

Eligibility Criteria

Eligible

You may qualify if you...

  • Healthy volunteers who understand the study and can give written consent
  • Male or female aged 18 to 55 years
  • Body mass index between 18 and 30 kg/m2
  • Weight at least 50.0 kg for males and 45.0 kg for females
  • Negative SARS-CoV-2 test on Day -2 (admission)
  • No significant medical history and in good health based on exams and lab tests
  • Females must be non-pregnant and non-lactating with negative pregnancy test
  • Willingness to use effective contraception from screening to 6 months after last dose
  • Willingness to avoid sperm or egg donation during study and 6 months after last dose
  • Willing and able to comply with study visits and procedures
Not Eligible

You will not qualify if you...

  • History of allergy including anaphylaxis to food, drugs, or any study drug component
  • Vegan diet or medical dietary restrictions
  • History of relevant respiratory, immune, skin, connective tissue, lymphatic, metabolic, liver, kidney, blood, lung, heart, digestive, muscle, urinary, hormone, nerve, psychiatric, or other disorders
  • Acute gastrointestinal symptoms at screening or admission (nausea, vomiting, diarrhea, heartburn)
  • Acute infections like influenza at screening or admission
  • Increased risk of infection, including tuberculosis history or positive TB test, residence in endemic regions, or unsafe sexual practices
  • Active cancer or cancer in last 5 years except superficial basal cell carcinoma
  • History suggesting abnormal immune function

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 1 location

1

Shanghai Xuhui Distric Central Hospital

Shanghai, China, 200031

Actively Recruiting

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Research Team

Q

Qian Chen, MD

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

QUADRUPLE

Allocation

RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

3

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A Single and Multiple Ascending Dose Trial of LT-002-158 Tablets in Healthy Adult Volunteers | DecenTrialz