Actively Recruiting

Phase 1
Age: 18Years +
MALE
NCT04221542

Study of AMG 509 in Participants With Metastatic Castration-Resistant Prostate Cancer

Led by Amgen · Updated on 2026-05-08

479

Participants Needed

57

Research Sites

628 weeks

Total Duration

On this page

Sponsors

A

Amgen

Lead Sponsor

B

BeiGene

Collaborating Sponsor

AI-Summary

What this Trial Is About

The overall aim of the trial is to evaluate the safety, tolerability, and pharmacokinetics (PK) of AMG 509 (monotherapy and in combination with abiraterone acetate and enzalutamide) and to evaluate preliminary efficacy. As of Protocol Amendment 10 (09 July 2025), only Parts 4A expansion, 6, and 7 are open to accrual.

CONDITIONS

Official Title

Study of AMG 509 in Participants With Metastatic Castration-Resistant Prostate Cancer

Who Can Participate

Age: 18Years +
MALE

Eligibility Criteria

Eligible

You may qualify if you...

  • Male participants aged 18 years or older
  • Histologically or cytologically confirmed metastatic castration-resistant prostate cancer
  • Refractory to or medically unsuitable for novel antiandrogen therapies including abiraterone acetate, enzalutamide, apalutamide, or darolutamide
  • Failed at least one but no more than two taxane chemotherapy regimens or refused taxane treatment
  • For dose-expansion phases, limited prior systemic anti-cancer treatments as specified
  • Underwent bilateral orchiectomy or on continuous androgen-deprivation therapy with GnRH agonist or antagonist
  • Total serum testosterone level of 50 ng/dL or less
  • Evidence of progressive disease by PSA, imaging, or bone scan criteria
  • Eastern Cooperative Oncology Group performance status of 0 or 1
  • Life expectancy of at least 3 months
  • Adequate organ function including hematological, renal, hepatic, cardiac, and pulmonary parameters as defined
  • For Part 3-Retreatment group: prior benefit from AMG 509 initial treatment and willingness to have fresh tumor biopsy if needed
Not Eligible

You will not qualify if you...

  • Presence of small cell or neuroendocrine prostate carcinoma or any histology other than adenocarcinoma
  • Radiation therapy within 4 weeks before first dose or local radiotherapy within 2 weeks
  • Untreated central nervous system metastases or leptomeningeal disease
  • Major surgery within 4 weeks before first dose
  • Active systemic infection within 7 days prior to treatment, except certain controlled infections
  • History or current autoimmune disease requiring permanent immunosuppressive therapy
  • Recent arterial thrombosis within 12 months or venous thrombosis within 6 months unless stable on anticoagulation
  • Myocardial infarction or symptomatic heart failure within 12 months, with some exceptions
  • Recent anti-cancer or immunotherapy within 4 weeks before first dose, excluding certain hormone therapies
  • Prior prostate specific membrane antigen radionuclide therapy within 2 months unless limited exposure
  • For Part 3-Retreatment: any anti-cancer therapy after last AMG 509 dose except certain hormone or bone therapies

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 57 locations

1

City of Hope National Medical Center

Duarte, California, United States, 91010

Actively Recruiting

2

Providence Saint Jude Medical Center

Fullerton, California, United States, 92835

Actively Recruiting

3

University of California San Francisco

San Francisco, California, United States, 94158

Actively Recruiting

4

Rocky Mountain Cancer Centers

Aurora, Colorado, United States, 80012

Actively Recruiting

5

Yale New Haven Hospital

New Haven, Connecticut, United States, 06520

Actively Recruiting

6

Emory University

Atlanta, Georgia, United States, 30322

Actively Recruiting

7

Indiana University

Indianapolis, Indiana, United States, 46202

Actively Recruiting

8

MidAmerica Cancer Care

Merriam, Kansas, United States, 66204

Actively Recruiting

9

Tulane Medical Center

New Orleans, Louisiana, United States, 70112

Completed

10

Washington University

St Louis, Missouri, United States, 63110

Actively Recruiting

11

Memorial Sloan Kettering Cancer Center

New York, New York, United States, 10065

Actively Recruiting

12

Duke University Medical Center Duke Cancer Center

Durham, North Carolina, United States, 27710

Actively Recruiting

13

Wake Forest University Health Sciences

Winston-Salem, North Carolina, United States, 27103

Actively Recruiting

14

Oncology Hematology Care Incorporated

Cincinnati, Ohio, United States, 45242

Actively Recruiting

15

Thomas Jefferson University

Philadelphia, Pennsylvania, United States, 19107

Actively Recruiting

16

University of Pittsburgh Medical Center

Pittsburgh, Pennsylvania, United States, 15232

Actively Recruiting

17

Prisma Health Upstate

Greenville, South Carolina, United States, 29605

Completed

18

Sanford Oncology Clinic and Pharmacy

Sioux Falls, South Dakota, United States, 57104

Actively Recruiting

19

United States Oncology Regulatory Affairs Corporate Office

Nashville, Tennessee, United States, 37203

Actively Recruiting

20

University of Texas MD Anderson Cancer Center

Houston, Texas, United States, 77030

Actively Recruiting

21

US Oncology Research Investigational Products Center

Irving, Texas, United States, 75063

Actively Recruiting

22

Intermountain Medical Center

Murray, Utah, United States, 84107

Actively Recruiting

23

Virginia Cancer Specialists PC

Fairfax, Virginia, United States, 22031

Actively Recruiting

24

Virginia Oncology Associates

Norfolk, Virginia, United States, 23502

Actively Recruiting

25

Fred Hutchinson Cancer Center

Seattle, Washington, United States, 98109

Actively Recruiting

26

Chris OBrien Lifehouse

Camperdown, New South Wales, Australia, 2050

Actively Recruiting

27

Monash Medical Centre

Clayton, Victoria, Australia, 3168

Actively Recruiting

28

Peking University First Hospital

Beijing, Beijing Municipality, China, 100034

Actively Recruiting

29

Sun Yat-sen University Cancer Center

Guangzhou, Guangdong, China, 510060

Actively Recruiting

30

The First Affiliated Hospital of Nanchang University

Nanchang, Jiangxi, China, 330006

Actively Recruiting

31

Fudan University Shanghai Cancer Centre

Shanghai, Shanghai Municipality, China, 200032

Actively Recruiting

32

Zhejiang Provincial Peoples Hospital

Hangzhou, Zhejiang, China, 314408

Actively Recruiting

33

Nanjing Drum Tower Hospital

Nanjing, China, 210003

Actively Recruiting

34

The First Affiliated Hospital of Wenzhou Medical University

Wenzhou, China, 325000

Actively Recruiting

35

Universitaetsklinikum Essen

Essen, Germany, 45147

Actively Recruiting

36

Universitaetsklinikum Heidelberg

Heidelberg, Germany, 69120

Actively Recruiting

37

Klinikum rechts der Isar der TUM

München, Germany, 81675

Actively Recruiting

38

Universitaetsklinikum Muenster

Münster, Germany, 48149

Actively Recruiting

39

National Cancer Center Hospital East

Kashiwa-shi, Chiba, Japan, 277-8577

Actively Recruiting

40

Yokohama City University Hospital

Yokohama, Kanagawa, Japan, 236-0004

Actively Recruiting

41

The Cancer Institute Hospital of Japanese Foundation for Cancer Research

Koto-ku, Tokyo, Japan, 135-8550

Actively Recruiting

42

Hospital da Luz, SA

Lisbon, Portugal, 1500-650

Actively Recruiting

43

Unidade Local de Saude de Santa Maria, EPE - Hospital de Santa Maria

Lisbon, Portugal, 1649-035

Actively Recruiting

44

Instituto Portugues de Oncologia do Porto Francisco Gentil, EPE

Porto, Portugal, 4200-072

Actively Recruiting

45

Seoul National University Hospital

Seoul, South Korea, 03080

Actively Recruiting

46

Asan Medical Center

Seoul, South Korea, 138-736

Actively Recruiting

47

Hospital Universitari Vall d Hebron

Barcelona, Catalonia, Spain, 08035

Actively Recruiting

48

Hospital Clinic i Provincial de Barcelona

Barcelona, Catalonia, Spain, 08036

Actively Recruiting

49

Clinica Universidad de Navarra

Pamplona, Navarre, Spain, 31008

Actively Recruiting

50

Hospital Clinico San Carlos

Madrid, Spain, 28040

Actively Recruiting

51

Hospital Universitario 12 de Octubre

Madrid, Spain, 28041

Actively Recruiting

52

Istituto Oncologico della Svizzera Italiana

Bellinzona, Switzerland, 6500

Actively Recruiting

53

Kantonsspital Graubuenden

Chur, Switzerland, 7000

Actively Recruiting

54

Centre Hospitalier Universitaire Vaudois

Lausanne, Switzerland, 1011

Actively Recruiting

55

Kantonsspital Sankt Gallen

Sankt Gallen, Switzerland, 9007

Actively Recruiting

56

National Taiwan University Hospital

Taipei, Taiwan, 10002

Actively Recruiting

57

Linkou Chang Gung Memorial Hospital of Chang Gung Medical Foundation

Taoyuan, Taiwan, 33305

Actively Recruiting

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Research Team

A

Amgen Call Center

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

7

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