Actively Recruiting

Phase 1
Age: 18Years - 130Years
All Genders
ID03423628

A Phase I, Multicenter Study to Assess the Safety, Tolerability, and Pharmacokinetics of Ascending Doses of AZD1390 in Combination With Radiation Therapy in Patients With Glioblastoma Multiforme and Brain Metastases from Solid Tumors

Led by AstraZeneca · Updated on 2025-12-22

180

Participants Needed

12

Research Sites

N/A

Total Duration

On this page

AI-Summary

What this Trial Is About

Researchers are evaluating the investigational drug AZD1390 combined with radiation therapy for treating brain tumors, including glioblastoma multiforme and brain metastases from solid tumors. This Phase 1, open-label study is the first to give AZD1390 to patients and aims to test the safety, tolerability, and how the drug is absorbed and processed in the body at increasing doses alongside different radiation therapy regimens. The study has three treatment arms with varying radiation schedules: Arm A uses 35 Gy of intensity-modulated radiation therapy (IMRT) over 2 weeks for recurrent glioblastoma; Arm B, now closed to recruitment, used 30 Gy of whole or partial brain radiation over 2 weeks for brain metastases; and Arm C uses 60 Gy of IMRT over 6 weeks for primary glioblastoma. AZD1390 is given in cycles before, during, and after radiation therapy, with some participants in Arm A undergoing an optional food effect assessment. Participants will undergo assessments including imaging scans every 8 weeks, blood tests to measure drug levels, and monitoring for side effects from treatment start until about 9 months after the last patient begins treatment. Researchers will track dose-limiting toxicities, adverse events, survival, and tumor response using established criteria. The study includes safety monitoring throughout and collects data on how the drug interacts with food in some participants.

CONDITIONS

Brief Title

A Study to Assess the Safety and Tolerability of AZD1390 Given With Radiation Therapy in Patients With Brain Cancer

Who Can Participate

Age: 18Years - 130Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Provision of formalin-fixed paraffin embedded tissue sample from primary or metastatic disease
  • Karnofsky Performance Score of 60 or higher
  • Histologically proven diagnosis of glioblastoma multiforme (GBM) or brain metastases as specified per arm
  • Radiological diagnosis of recurrent, relapsed, or progressive disease according to RANO criteria for Arm A
  • Completion of first-line radiation at least 6 months prior to treatment start for Arm A
  • Well controlled tumor-induced seizures and willingness to receive anti-epileptic prophylaxis during study drug administration
  • Histologically proven solid tumor malignancy with brain lesions for Arm B (closed to recruitment)
  • No prior brain radiation to the treatment area for Arm B
  • Histologically proven primary GBM with unmethylated MGMT promoter status and IDH1 mutational testing for Arm C
  • No history of uncontrolled seizures after surgery for Arm C
  • Specific fasting and dietary requirements for optional food effect assessment in Arm A
Not Eligible

You will not qualify if you...

  • Chemotherapy or investigational drugs within 28 days prior to treatment start, or carmustine/lomustine within 6 weeks for Arms A and C
  • Checkpoint inhibitors within 28 days prior to treatment start and other agents within 7 days for Arm B
  • History of severe brain injury or stroke
  • Inability to undergo sequential MRI evaluations
  • History of epileptic disorder or seizures unrelated to tumor
  • Treatment with strong CYP3A4 inhibitors or inducers within 2 weeks prior to study drug
  • Concurrent use of seizurogenic medications
  • History or presence of interstitial lung disease, drug-induced ILD, or radiation pneumonitis requiring steroids
  • Severe or uncontrolled medical conditions such as COPD
  • Prior pneumotoxic drug treatment within the past year with lung toxicity
  • History or presence of myopathy or elevated creatine kinase greater than 5 times upper limit of normal
  • Cardiac dysfunction including recent myocardial infarction or unstable angina
  • Active severe pulmonary infections (specific to Japan part)
  • Unresolved toxicities greater than grade 1 except alopecia
  • Prior treatment with ATM inhibitor with concurrent radiation for Arm A and Japan part
  • Diabetes or systemic steroid treatment for food effect assessment in Arm A (not applicable in Japan part)

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

1
2
3
+1

Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person)

Treatment

Duration - 2 weeks for Arm A and B; 6 weeks for Arm C

Participants receive AZD1390 in combination with radiation therapy according to their assigned arm. Treatment includes up to 3 cycles of AZD1390 dosing and radiation therapy that varies by arm.

Daily visits for radiation therapy over the treatment period plus dosing visits for AZD1390

Follow-up

Duration - Up to 9 months for Arms A and C; approximately 8 weeks for Arm B

Participants are monitored for safety, tolerability, and response after completion of treatment. Follow-up includes assessments over approximately 9 months for Arms A and C and about 8 weeks for Arm B.

Regular visits approximately every 8 weeks for response assessments starting 4 weeks after radiation therapy

Trial Site Locations

Total: 12 locations

1

Research Site

Boston, Massachusetts, United States, 02114

Actively Recruiting

2

Research Site

Boston, Massachusetts, United States, 02215

Actively Recruiting

3

Research Site

New York, New York, United States, 10065

Actively Recruiting

4

Research Site

Pittsburgh, Pennsylvania, United States, 15232

Actively Recruiting

5

Research Site

Richmond, Virginia, United States, 23298

Actively Recruiting

6

Research Site

Chūōku, Japan, 104-0045

Completed

7

Research Site

Hidaka-shi, Japan, 350-1298

Active, Not Recruiting

8

Research Site

Kyoto, Japan, 606-8507

Active, Not Recruiting

9

Research Site

Cambridge, United Kingdom, CB2 0QQ

Active, Not Recruiting

10

Research Site

Glasgow, United Kingdom, G12 0YN

Completed

11

Research Site

Leeds, United Kingdom, LS9 7TF

Actively Recruiting

12

Research Site

London, United Kingdom, W1T 7HA

Withdrawn

Loading map...

Research Team

A

AstraZeneca Clinical Study Information Center

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

3

Similar Trials

Exploring the Feasibility of Cerebrospinal Fluid Liquid Biop...

Solid Tumor Malignancies

Actively Recruiting

1 location

Frequently Asked Questions

Have more questions? Get in touch with our team for quick support

Not the Right Trial for You?

Explore thousands of other clinical trials that might be a better match.
Sign up to get personalized trial recommendations delivered to your inbox.

Already have an account? Log in here