Actively Recruiting

Phase 1
Age: 40Years - 80Years
All Genders
ID07214727

A Phase 1, Randomized, Placebo-Controlled Study With Double-Blind and Open-Label Extension Periods to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of Intrathecal ALN-5288 in Adults With Alzheimer's Disease

Led by Alnylam Pharmaceuticals · Updated on 2026-05-14

50

Participants Needed

13

Research Sites

N/A

Total Duration

On this page

Sponsors

A

Alnylam Pharmaceuticals

Lead Sponsor

R

Regeneron Pharmaceuticals

Collaborating Sponsor

AI-Summary

What this Trial Is About

Researchers are evaluating the safety and tolerability of a drug called ALN-5288, given through a spinal injection, in adults aged 40 to 80 with Alzheimer's Disease (AD). This Phase 1 randomized study also examines how the body processes ALN-5288 and its effects after dosing. Participants have mild cognitive impairment or dementia due to AD, confirmed by specific brain scans or cerebrospinal fluid tests within seven years before screening. Participants are randomly assigned to receive either ALN-5288 or a placebo during the double-blind period. After this, all participants receive ALN-5288 in an open-label extension phase. Both ALN-5288 and placebo are administered intrathecally (into the spinal fluid). The study tracks participants for up to 32 months from the first dose to monitor treatment effects and safety. During the study, participants undergo regular assessments including monitoring of any adverse events, blood and urine tests to measure ALN-5288 levels, and cerebrospinal fluid tests to evaluate biomarkers related to Alzheimer's Disease. Researchers carefully observe the frequency and severity of any side effects. The study aims to gather detailed information on how the drug behaves in the body and its impact, while ensuring participant safety over the long follow-up period.

CONDITIONS

Brief Title

A Study to Evaluate ALN-5288 in Patients With Alzheimer's Disease

Who Can Participate

Age: 40Years - 80Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Able and willing to meet all study requirements as judged by the Investigator
  • Diagnosed with Alzheimer's disease based on clinical findings supported by cerebrospinal fluid biomarkers or positive PET amyloid imaging within 7 years before screening
  • Has mild cognitive impairment or dementia due to Alzheimer's disease
  • Age between 40 and 80 years
Not Eligible

You will not qualify if you...

  • Diagnosed with non-Alzheimer's dementia
  • Alanine aminotransferase (ALT) or aspartate aminotransferase (AST) levels greater than 2 times the upper limit of normal
  • Total bilirubin greater than 1.5 times the upper limit of normal
  • Known HIV infection
  • History of hepatitis C or current hepatitis B infection
  • Systolic blood pressure over 160 mmHg or diastolic blood pressure over 100 mmHg after 10 minutes rest at screening
  • Estimated glomerular filtration rate (eGFR) less than 45 mL/min/1.73 m² at screening
  • Clinically significant ECG abnormalities at screening
  • Uncontrolled psychiatric conditions including high suicide risk, major depression, psychosis, confusion, or violent behavior
  • History of bleeding disorders due to chronic conditions
  • Medical history of brain or spinal diseases interfering with spinal injection and lumbar puncture
  • Uncontrolled seizures within the last 6 months prior to screening

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person)

Treatment

Duration - Up to 32 months

Participants receive intrathecal administration of ALN-5288 or placebo during the double-blind period, followed by open-label extension where all participants receive ALN-5288.

Regular visits during both double-blind and open-label extension periods

Trial Site Locations

Total: 13 locations

1

Clinical Trial Site

Montreal, Canada, H3G 1H9

Actively Recruiting

2

Clinical Trial Site

Ottawa, Canada, K1Z 1G3

Actively Recruiting

3

Clinical Trial Site

Toronto, Canada, M3B 2S7

Actively Recruiting

4

Clinical Trial Site

Toronto, Canada, M5T 2S8

Not Yet Recruiting

5

Clinical Trial Site

's-Hertogenbosch, Netherlands, 5223

Not Yet Recruiting

6

Clinical Trial Site

Amsterdam, Netherlands, 1081 GN

Not Yet Recruiting

7

Clinical Trial Site

Barcelona, Spain, 08036

Not Yet Recruiting

8

Clinical Trial Site

Madrid, Spain, 28040

Not Yet Recruiting

9

Clinical Trial Site

Sant Cugat del Vallès, Spain, 08190

Not Yet Recruiting

10

Clinical Trial Site

Glasgow, United Kingdom, G51 4TF

Not Yet Recruiting

11

Clinical Trial Site

London, United Kingdom, WC1N 3BG

Actively Recruiting

12

Clinical Trial Site

Sheffield, United Kingdom, S10 2JF

Not Yet Recruiting

13

Clinical Trial Site

Southampton, United Kingdom, SO16 6YD

Not Yet Recruiting

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Research Team

C

Clinical Trial Information Line

C

Clinical Trial Information Line

How is the study designed?

Study Type

INTERVENTIONAL

Masking

TRIPLE

Allocation

RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

2

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