Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT04953897

Study to Evaluate the Pharmacokinetics and Safety of Oral Decitabine and Cedazuridine in Cancer Patients With Renal Impairment

Led by Taiho Oncology, Inc. · Updated on 2026-04-30

18

Participants Needed

21

Research Sites

258 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

This is a Phase 1b, multicenter, open-label, PK, and safety study of multiple oral doses of oral decitabine and cedazuridine (formerly known as ASTX727) as a fixed-dose combination of decitabine 35 milligrams (mg) and cedazuridine 100 mg in cancer participants with severe renal impairment and cancer participants with normal renal function as matched control participants. Adult participants with acute myeloid lymphoma (AML), myelodysplastic syndrome (MDS), or solid tumors who are candidates to receive oral decitabine and cedazuridine will be enrolled in this study. Study duration per participant is approximately up to 8 weeks.

CONDITIONS

Official Title

Study to Evaluate the Pharmacokinetics and Safety of Oral Decitabine and Cedazuridine in Cancer Patients With Renal Impairment

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Able to understand and comply with study procedures and provide informed consent
  • Histologically or cytologically confirmed malignancy: metastatic or unresectable solid tumor without standard life-prolonging options, or AML, MDS, or other hematologic malignancy without standard life-prolonging options
  • For AML/MDS: confirmed diagnosis except M3 acute promyelocytic leukemia, or frontline MDS/treatment-naive AML not suitable for induction therapy
  • Platelet count ≥25,000/μL and absolute neutrophil count (ANC) ≥100 cells/μL for AML/MDS; platelet count ≥100,000/μL and ANC ≥1000 cells/μL for other hematologic malignancies or solid tumors
  • Eastern Cooperative Oncology Group (ECOG) performance status 0 to 3
  • Adequate liver function: total or direct bilirubin ≤1.5 times upper limit of normal (ULN); AST and ALT ≤2.5 times ULN
  • Stable creatinine clearance (CLcr) by Cockcroft-Gault equation: ≥80 mL/min/1.73m² for normal renal function group or <30 mL/min/1.73m² for severe renal impairment group (without dialysis), with less than 30% deviation from screening to baseline
  • No major surgery within 30 days before first dose
  • Life expectancy of at least 3 months
  • Women of childbearing potential must not be pregnant or breastfeeding and must have a negative pregnancy test
  • Women of childbearing potential must agree to use highly effective contraception during and for 6 months after treatment
  • Male participants with female partners of childbearing potential must use condoms and recommend contraception to partners during and for 3 months after treatment
Not Eligible

You will not qualify if you...

  • Treatment with azacitidine or decitabine within 4 weeks before screening
  • Prior cytotoxic chemotherapy for AML except hydroxyurea for high white blood cell counts
  • Hospitalization for febrile neutropenia, pneumonia, sepsis, or systemic infection longer than 2 days within 30 days before first dose
  • Treatment with investigational or other cancer therapies within 2 weeks or 5 half-lives before first dose, or ongoing adverse events from prior treatments
  • Concurrent myelodysplastic syndrome therapies unless completed at least 1 week before first dose
  • Live vaccines within 4 weeks before first dose until after follow-up visit
  • High medical risk due to uncontrolled systemic diseases or infections
  • Conditions causing QT prolongation or history of torsades de pointes
  • Unstable heart disease or severe heart failure, uncontrolled hypertension or significant hypotension
  • Significant mental illness or substance abuse risking noncompliance
  • Rapidly progressive or highly proliferative AML/MDS at high risk for intensive chemotherapy within 3 months
  • Life-threatening illness or severe organ dysfunction compromising safety or study completion
  • Untreated central nervous system metastases; treated metastases must be stable for at least 4 weeks
  • Infection with HIV or active hepatitis B or C
  • History of alcohol abuse or drug addiction
  • Excessive alcohol consumption above specified weekly limits
  • Blood donation or loss over 500 mL within 60 days before first dose
  • Hypersensitivity to study drugs or excipients

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 21 locations

1

MD Anderson

Houston, Texas, United States, 77030

Actively Recruiting

2

Erebuni Medical Center

Yerevan, Armenia

Actively Recruiting

3

Hematology Center After Prof. R. Yeolyan (Adult Blood Disorders)

Yerevan, Armenia

Actively Recruiting

4

Hematology Center After Prof. R. Yeolyan (Clinic of Adults Oncology)

Yerevan, Armenia

Actively Recruiting

5

National Center of Oncology Named After V.A. Fanarjyan

Yerevan, Armenia

Actively Recruiting

6

Complex Oncology Center - Plovdiv - Base II

Plovdiv, Bulgaria

Withdrawn

7

BIO1

Vilnius, Lithuania

Withdrawn

8

Centrum Badań Klinicznych Piotr Napora Lekarze Sp. p.

Wroclaw, Poland, 51-162

Actively Recruiting

9

Institutul Oncologic Bucuresti - Prof. Dr. Alexandru Trestioreanu

Bucharest, Romania, 22328

Actively Recruiting

10

Institutul Oncologic Prof. Dr. Ion Chiricuta

Cluj-Napoca, Romania, 400015

Actively Recruiting

11

Summit Clinical Research s.r.o

Bratislava, Slovakia, 831 01

Actively Recruiting

12

START Barcelona - Hospital HM Nou Delfos

Barcelona, Spain, 8023

Actively Recruiting

13

Hospital Universitari Dexeus - Grupo Quirónsalud

Barcelona, Spain

Withdrawn

14

START Rioja - Hospital de San Pedro

La Rioja, Spain, 26006

Not Yet Recruiting

15

Hospital Universitari Arnau de Vilanova

Lleida, Spain

Actively Recruiting

16

START Madrid - Hospital Universitario Fundación Jiménez Díaz

Madrid, Spain, 28040

Actively Recruiting

17

START Madrid - CIOCC - HM Sanchinarro

Madrid, Spain, 28050

Actively Recruiting

18

Hospital Universitario 12 de Octubre

Madrid, Spain

Withdrawn

19

Hospital Clínico Universitario Virgen de la Arrixaca (Hematology Dept)

Murcia, Spain, 30120

Actively Recruiting

20

Hospital Clínico Universitario Virgen de la Arrixaca (Solid Tumor Dept)

Murcia, Spain

Actively Recruiting

21

Hospital Universitari i Politècnic La Fe

Valencia, Spain

Terminated

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Research Team

T

Taiho Oncology, Inc.

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

2

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