Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT04953910

Study to Evaluate the Pharmacokinetics and Safety of Oral Decitabine and Cedazuridine in Cancer Patients With Hepatic Impairment

Led by Taiho Oncology, Inc. · Updated on 2026-04-30

27

Participants Needed

22

Research Sites

205 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

This is a Phase 1b, multicenter, open-label, pharmacokinetic (PK), and safety study of multiple oral doses of oral decitabine and cedazuridine (formerly known as ASTX727) as a fixed-dose combination of decitabine 35 milligrams (mg) and cedazuridine 100 mg in cancer participants with moderate and severe hepatic impairment and cancer participants with normal hepatic function as control participants. Participants with severe hepatic impairment will be enrolled only after the safety evaluation of at least 6 participants with moderate hepatic impairment has been determined and supports the enrollment of participants with severe hepatic impairment. Adult participants with acute myeloid lymphoma (AML), myelodysplastic syndrome (MDS), or solid tumors who are candidates to receive oral decitabine and cedazuridine will be enrolled in this study. Study duration is per participant approximately up to 8 weeks.

CONDITIONS

Official Title

Study to Evaluate the Pharmacokinetics and Safety of Oral Decitabine and Cedazuridine in Cancer Patients With Hepatic Impairment

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Able to understand and comply with study procedures and provide informed consent
  • Have a confirmed diagnosis of metastatic or unresectable solid tumor without standard life-prolonging options, or diagnosis of AML or MDS, or other hematologic malignancy without standard life-prolonging options
  • For AML/MDS participants: confirmed diagnosis per 2008 WHO classification, or frontline MDS/treatment-naive AML not suitable for induction therapy
  • Platelet count \u226525,000 per microliter and absolute neutrophil count \u2265100 cells/\u03bcL for AML/MDS participants
  • For other hematologic malignancies or solid tumors: platelet count \u2265100,000/\u03bcL and ANC \u22651000 cells/\u03bcL
  • ECOG performance status between 0 and 3
  • Hepatic function classified as normal, moderate impairment, or severe impairment per NCI CTEP criteria
  • Adequate kidney function with creatinine clearance over 50 mL/min
  • No major surgery within 30 days before first drug dose
  • Life expectancy of at least 3 months
  • Women of childbearing potential must not be pregnant or breastfeeding, must have negative pregnancy test, and agree to use effective contraception
  • Male participants with female partners of childbearing potential must agree to use condoms and advise partner to use effective contraception
Not Eligible

You will not qualify if you...

  • Treatment with azacitidine or decitabine within 4 weeks before screening
  • Recent hospitalization over 2 days for febrile neutropenia, pneumonia, sepsis, or systemic infection within 30 days before first dose
  • Treatment with investigational or other cancer therapies within 2 weeks or 5 half-lives before first dose, or ongoing adverse events from prior treatment
  • Concurrent MDS therapies except certain short-term uses approved by physician
  • Administration of live vaccines within 4 weeks before first dose until after follow-up
  • High medical risk from uncontrolled diseases, infections, or comorbidities
  • Conditions causing prolonged QT interval or history of dangerous heart rhythms
  • Unstable heart disease or uncontrolled hypertension
  • Significant mental illness or substance abuse that risks noncompliance
  • Rapidly progressing AML/MDS or high risk for intensive chemotherapy within 3 months
  • Life-threatening illness or severe organ dysfunction affecting safety or study completion
  • Untreated CNS metastases; treated metastases must be stable for at least 4 weeks
  • HIV infection
  • Active hepatitis C infection (HCV+ with positive RNA PCR)
  • Active hepatitis B infection (HBsAg+)
  • Excessive alcohol consumption (over 24 units/week for males, 17 units/week for females)
  • Recent blood donation or loss over 500 mL within 60 days before first dose
  • Allergy to decitabine, cedazuridine, or their ingredients

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 22 locations

1

MD Anderson

Houston, Texas, United States, 77030

Actively Recruiting

2

Erebuni Medical Center

Yerevan, Armenia

Actively Recruiting

3

Hematology Center After Prof. R. Yeolyan (Adult Blood Disorders)

Yerevan, Armenia

Actively Recruiting

4

Hematology Center After Prof. R. Yeolyan (Clinic of Adults Oncology)

Yerevan, Armenia

Actively Recruiting

5

National Center of Oncology Named After V.A. Fanarjyan

Yerevan, Armenia

Actively Recruiting

6

Complex Oncology Center - Plovdiv - Base II

Plovdiv, Bulgaria

Withdrawn

7

BIO1

Vilnius, Lithuania

Withdrawn

8

Centrum Badań Klinicznych Piotr Napora Lekarze Sp. p.

Wroclaw, Poland, 51-162

Actively Recruiting

9

Institutul Oncologic Bucuresti - Prof. Dr. Alexandru Trestioreanu

Bucharest, Romania, 22328

Actively Recruiting

10

Institutul Oncologic Prof. Dr. Ion Chiricuta

Cluj-Napoca, Romania, 400015

Actively Recruiting

11

Summit Clinical Research s.r.o

Bratislava, Slovakia, 831 01

Actively Recruiting

12

START Barcelona - Hospital HM Nou Delfos

Barcelona, Spain, 8023

Actively Recruiting

13

Hospital Universitari Dexeus - Grupo Quirónsalud

Barcelona, Spain

Withdrawn

14

START Rioja - Hospital de San Pedro

La Rioja, Spain, 26006

Not Yet Recruiting

15

Hospital Universitari Arnau de Vilanova

Lleida, Spain

Actively Recruiting

16

START Madrid - Hospital Universitario Fundación Jiménez Díaz

Madrid, Spain, 28040

Actively Recruiting

17

Hospital Universitario La Paz

Madrid, Spain, 28046

Actively Recruiting

18

START Madrid - CIOCC - HM Sanchinarro

Madrid, Spain, 28050

Actively Recruiting

19

Hospital Universitario 12 de Octubre

Madrid, Spain

Withdrawn

20

Hospital Clínico Universitario Virgen de la Arrixaca (Hematology Dept)

Murcia, Spain, 30120

Actively Recruiting

21

Hospital Clínico Universitario Virgen de la Arrixaca (Solid Tumor Dept)

Murcia, Spain

Actively Recruiting

22

Hospital Universitari i Politècnic La Fe

Valencia, Spain

Terminated

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Research Team

T

Taiho Oncology, Inc.

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

3

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Study to Evaluate the Pharmacokinetics and Safety of Oral Decitabine and Cedazuridine in Cancer Patients With Hepatic Impairment | DecenTrialz