Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT06431594

A Study to Evaluate the Safety, Tolerability, Pharmacokinetics and Clinical Activity of GSK5733584 for Injection in Participants With Advanced Solid Tumors

Led by GlaxoSmithKline · Updated on 2025-06-25

385

Participants Needed

47

Research Sites

167 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

The goal of this study is to assess the safety and tolerability of GSK5733584. The study will also see how the levels of GSK5733584 change over time at different dose amount.

CONDITIONS

Official Title

A Study to Evaluate the Safety, Tolerability, Pharmacokinetics and Clinical Activity of GSK5733584 for Injection in Participants With Advanced Solid Tumors

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Males or females aged 18 years or older (≥18 years)
  • Participants with pathologically confirmed advanced solid tumor who have failed or are intolerant to standard of care
  • Histologically documented advanced (metastatic and/or unresectable) high-grade serous/endometrioid ovarian, primary peritoneal, or fallopian tube cancer for PROC cohort
  • Received or intolerant to 1 to 3 lines of prior systemic therapy
  • Platinum-resistant disease defined as progression or relapse within 6 months after platinum-based therapy
  • Prior bevacizumab if considered a candidate and locally available
  • Known Folate receptor-α expressing tumors must have received mirvetuximab soravtasine if candidate and locally available
  • Known BRCA mutated tumors should have received a PARP inhibitor if candidate and locally available
  • Histologically documented advanced or recurrent endometrial cancer for endometrial cancer cohort
  • Received or intolerant to 1 to 3 lines of prior systemic therapy
  • Prior platinum and PD(L)-1 inhibitor if candidate and locally available
  • All epithelial histologies including carcinosarcoma permitted
  • At least one target lesion per RECIST 1.1
  • Tumor tissue from new biopsy or archival tissue within 2 years prior to first dose for biomarker analysis
  • ECOG Performance Status of 0 to 2 with no deterioration within 2 weeks before first dose
  • Life expectancy of at least 12 weeks
Not Eligible

You will not qualify if you...

  • Received any B7-H4-targeted therapies
  • Received cytotoxic chemotherapy, anti-tumor traditional Chinese medicines, or other anti-tumor drugs within 28 days prior to first dose or need to continue during study
  • Received locoregional radiation therapy within 2 weeks prior to first dose
  • More than 30% bone marrow irradiation or wide-field radiation therapy within 4 weeks prior to first dose
  • Presence of pleural or abdominal effusion or ascites requiring intervention; presence of pericardial effusion
  • Major surgery within 28 days prior to first dose
  • Evidence of brain metastasis unless asymptomatic
  • Inadequate bone marrow reserve or hepatic/renal functions
  • Mean QTcF > 470 msec on resting ECG
  • Current clinically significant arrhythmias or ECG abnormalities
  • Risk factors for prolonged QTc or arrhythmia events
  • Left ventricular ejection fraction < 50%
  • Severe, uncontrolled or active cardiovascular disorders, serious or poorly controlled hypertension, clinically significant bleeding symptoms, or serious thromboembolic events
  • Current or prior interstitial lung disease or pneumonitis requiring high-dose systemic glucocorticoids
  • Prior therapy with topoisomerase inhibitors or topoisomerase inhibitor antibody-drug conjugates
  • For PROC cohort: primary platinum refractory disease (progression within 12 weeks of first line platinum therapy) not permitted
  • Non-epithelial carcinoma, clear-cell, mucinous, germ-cell, low-grade serous, or low-grade endometrioid carcinoma not permitted
  • For endometrial cancer: mesenchymal tumors of the uterus (uterine sarcomas) not permitted

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 47 locations

1

GSK Investigational Site

Lake Mary, Florida, United States, 32746

Actively Recruiting

2

GSK Investigational Site

Fairway, Kansas, United States, 66205

Actively Recruiting

3

GSK Investigational Site

Boston, Massachusetts, United States, 02114

Actively Recruiting

4

GSK Investigational Site

Boston, Massachusetts, United States, 02215

Actively Recruiting

5

GSK Investigational Site

Detroit, Michigan, United States, 48201

Actively Recruiting

6

GSK Investigational Site

Grand Rapids, Michigan, United States, 49546

Actively Recruiting

7

GSK Investigational Site

Nashville, Tennessee, United States, 37203

Actively Recruiting

8

GSK Investigational Site

Dallas, Texas, United States, 75230

Actively Recruiting

9

GSK Investigational Site

West Valley City, Utah, United States, 84119

Actively Recruiting

10

GSK Investigational Site

Cipoletti Rio Negro, Argentina, R8324CVE

Actively Recruiting

11

GSK Investigational Site

Ciudad de Buenos Aires, Argentina, 1118

Actively Recruiting

12

GSK Investigational Site

Rosario, Argentina, S2002

Actively Recruiting

13

GSK Investigational Site

Blacktown, New South Wales, Australia, 2148

Actively Recruiting

14

GSK Investigational Site

Macquarie University, New South Wales, Australia, 2109

Actively Recruiting

15

GSK Investigational Site

Leuven, Belgium, 3000

Actively Recruiting

16

GSK Investigational Site

Ottawa, Ontario, Canada, K1H 8L6

Actively Recruiting

17

GSK Investigational Site

Toronto, Ontario, Canada, M5G 2M9

Actively Recruiting

18

GSK Investigational Site

Montreal, Quebec, Canada, H2X 0A9

Actively Recruiting

19

GSK Investigational Site

Helsinki, Finland, 00180

Actively Recruiting

20

GSK Investigational Site

Helsinki, Finland, 00290

Actively Recruiting

21

GSK Investigational Site

Tampere, Finland, 33520

Actively Recruiting

22

GSK Investigational Site

Lyon, France, 69373

Actively Recruiting

23

GSK Investigational Site

Saint-Herblain, France, 44805

Actively Recruiting

24

GSK Investigational Site

Villejuif, France, 94805

Actively Recruiting

25

GSK Investigational Site

Roma, Italy, 00168

Actively Recruiting

26

GSK Investigational Site

Rozzano MI, Italy, 20089

Actively Recruiting

27

GSK Investigational Site

Saitama, Japan, 350-1298

Actively Recruiting

28

GSK Investigational Site

Shizuoka, Japan, 411-8777

Actively Recruiting

29

GSK Investigational Site

Tokyo, Japan, 135-8550

Actively Recruiting

30

GSK Investigational Site

Amsterdam, Netherlands, 1066 CX

Actively Recruiting

31

GSK Investigational Site

Gyeonggi-do, South Korea, 10408

Actively Recruiting

32

GSK Investigational Site

Seoul, South Korea, 03080

Actively Recruiting

33

GSK Investigational Site

Seoul, South Korea, 03722

Actively Recruiting

34

GSK Investigational Site

Seoul, South Korea, 06351

Actively Recruiting

35

GSK Investigational Site

Barcelona, Spain, 08035

Actively Recruiting

36

GSK Investigational Site

Córdoba, Spain, 14004

Actively Recruiting

37

GSK Investigational Site

Girona, Spain, 17007

Actively Recruiting

38

GSK Investigational Site

Madrid, Spain, 28027

Actively Recruiting

39

GSK Investigational Site

Madrid, Spain, 28034

Actively Recruiting

40

GSK Investigational Site

Madrid, Spain, 28040

Actively Recruiting

41

GSK Investigational Site

Madrid, Spain, 28046

Actively Recruiting

42

GSK Investigational Site

Pozuelo de AlarcOn Madr, Spain, 28223

Actively Recruiting

43

GSK Investigational Site

Stockholm, Sweden, 17164

Actively Recruiting

44

GSK Investigational Site

Uppsala, Sweden, SE-751 85

Actively Recruiting

45

GSK Investigational Site

Cambridge, United Kingdom, CB2 0QQ

Actively Recruiting

46

GSK Investigational Site

London, United Kingdom, NW1 2PG

Actively Recruiting

47

GSK Investigational Site

London, United Kingdom, W1G 6AD

Actively Recruiting

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Research Team

U

US GSK Clinical Trials Call Center

CONTACT

E

EU GSK Clinical Trials Call Center

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

2

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A Study to Evaluate the Safety, Tolerability, Pharmacokinetics and Clinical Activity of GSK5733584 for Injection in Participants With Advanced Solid Tumors | DecenTrialz