Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT05929235

A Study of FX-909 in Patients With Advanced Solid Malignancies, Including Advanced Urothelial Carcinoma

Led by Flare Therapeutics Inc. · Updated on 2026-04-20

120

Participants Needed

12

Research Sites

231 weeks

Total Duration

On this page

Sponsors

F

Flare Therapeutics Inc.

Lead Sponsor

M

Merck Sharp & Dohme LLC

Collaborating Sponsor

AI-Summary

What this Trial Is About

The goal of this clinical trial is to study the safety and tolerability in all advanced solid tumors, including advanced urothelial carcinoma. The main question\[s\] it aims to answer are: * Is FX-909 safe and tolerable, as a monotherapy and in combination with Pembrolizumab * What is the right dose level for patients Participants will be asked to take FX-909 daily in tablet form, or FX-909 daily and Pembrolizumab every 3 weeks, and record any outcomes from taking the drug. Participants will also be asked to return for multiple site visits for various blood tests and to collect blood and tumor samples as well as have regular CT/MRI scans.

CONDITIONS

Official Title

A Study of FX-909 in Patients With Advanced Solid Malignancies, Including Advanced Urothelial Carcinoma

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Able to understand and willing to sign an informed consent.
  • Age 18 years or older.
  • ECOG performance status 0, 1, or 2.
  • Provide an archival tumor sample no older than 30 months or consent to a fresh biopsy.
  • Part A: Diagnosed with locally advanced or metastatic solid tumors that progressed after or lack standard therapy.
  • Part B: Diagnosed with locally advanced or metastatic urothelial carcinoma with high PPARG expression (TPS  60%).
  • Treated with 4 or fewer prior therapies for advanced or metastatic disease.
  • Part A: Patients with or without measurable disease.
  • Part B: Patients with measurable disease per RECIST 1.1 not previously irradiated or progressed after radiation.
  • Meet required screening laboratory values.
  • For Part 1A1: ECOG 0 or 1, progressed after standard therapies including anti-PD-1/L1 treatment.
  • Provide archival or fresh tumor biopsy within 30 months.
  • Recovery from prior anticancer therapy adverse events to Grade 1 or baseline.
  • Males agree to use contraception during and 90 days after treatment.
  • Females of childbearing potential have negative pregnancy test and use contraception during and 120 days after treatment.
  • HIV-infected patients must have well-controlled HIV on ART.
  • Patients with controlled HBV or cured HCV infection.
  • Adequate organ function as defined in study tables.
Not Eligible

You will not qualify if you...

  • Pregnant or breastfeeding females.
  • Recent anticancer therapy within 2 weeks or 5 half-lives before study drug.
  • Prior therapy inhibiting PPARG or RXRA.
  • Unresolved adverse events from prior therapies above Grade 1.
  • Major surgery within 4 weeks before study drug.
  • Recent radiation therapy without adequate washout.
  • History of other malignancies within 2 years unless cured.
  • QTcF > 470 msec or history of long QT syndrome.
  • Active lipodystrophy/lipoatrophy or medications causing it.
  • Active infections requiring treatment.
  • Known HIV positive without viral suppression.
  • Active hepatitis B or C infection without control.
  • Recent pancreatitis or significant lung impairment.
  • Uncontrolled CNS metastases or leptomeningeal disease.
  • Need for high dose steroids or prohibited therapies.
  • Participation in other investigational studies.
  • Serious cardiovascular diseases or events within 6 months.
  • Recent thromboembolic or bleeding disorders.
  • Severe hypersensitivity to study drugs.
  • Gastrointestinal disorders affecting drug intake.
  • Family members involved in study staff unless approved.
  • Conditions hampering study compliance or safety.
  • Type 1 diabetes or uncontrolled type 2 diabetes requiring insulin.
  • Psychological or social conditions interfering with participation.

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 12 locations

1

UCSF Helen Diller Family Comprehensive Cancer Center

San Francisco, California, United States, 94158

Actively Recruiting

2

Yale Cancer Center

New Haven, Connecticut, United States, 06519

Actively Recruiting

3

Sylvester Comprehensive Cancer Center, University of Miami

Miami, Florida, United States, 33136

Actively Recruiting

4

The University of Chicago Medicine

Chicago, Illinois, United States, 60637

Actively Recruiting

5

Mass General Cancer Center

Boston, Massachusetts, United States, 02114

Actively Recruiting

6

Dana Farber Cancer Institute

Boston, Massachusetts, United States, 02215

Actively Recruiting

7

Icahn School of Medicine at Mount Sinai

New York, New York, United States, 10029

Actively Recruiting

8

Memorial Slone Kettering Cancer Center

New York, New York, United States, 10065

Actively Recruiting

9

UNC Lineberger Comprehensive Cancer Center

Chapel Hill, North Carolina, United States, 27514

Actively Recruiting

10

The Cleveland Clinic Foundation

Cleveland, Ohio, United States, 44195

Actively Recruiting

11

Sarah Cannon Research Institute

Nashville, Tennessee, United States, 37203

Actively Recruiting

12

Houston Methodist Cockrell Center for Advanced Therapeutics

Houston, Texas, United States, 77030

Actively Recruiting

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Research Team

J

Janine Koucheki, Associate Director, Clinical Operations

CONTACT

C

Carolyn McCrone, Sr Clinical Trial Associate

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

3

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