Actively Recruiting

Phase 1
Age: 18Years +
All Genders
NCT05853367

Study of MK-0472 in Participants With Advanced/Metastatic Solid Tumors (MK-0472-001)

Led by Merck Sharp & Dohme LLC · Updated on 2026-03-13

178

Participants Needed

25

Research Sites

240 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

The purpose of this study is to assess the efficacy, safety, and tolerability of MK-0472 administered as monotherapy and in combination with pembrolizumab (MK-3475) or MK-1084 in participants with histologically or cytologically confirmed diagnosis of advanced/metastatic solid tumors.

CONDITIONS

Official Title

Study of MK-0472 in Participants With Advanced/Metastatic Solid Tumors (MK-0472-001)

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Has histologically or cytologically confirmed advanced or metastatic solid tumor
  • Hepatitis B surface antigen (HBsAg) positive participants must have received antiviral therapy for at least 4 weeks and have undetectable HBV viral load before enrollment
  • Participants with history of hepatitis C virus (HCV) infection must have undetectable HCV viral load at screening
  • Participants with HIV must have well-controlled HIV on stable antiretroviral therapy for more than 4 weeks
  • Arm 1: Oncogenic receptor tyrosine kinase (RTK) pathway alterations confirmed and have received or been intolerant to all available beneficial treatments
  • Arm 2: Tumor types sensitive to anti-PD-1/L1 therapies including melanoma, NSCLC without EGFR/ALK/ROS1 mutations, renal cell carcinoma, urothelial carcinoma, Merkel cell carcinoma, MSI-high CRC, endometrial cancer, cervical cancer, small cell lung cancer, triple negative breast cancer, esophageal cancer, gastric cancer, biliary tract cancer, hepatocellular carcinoma, head and neck squamous cancer, cutaneous squamous cancer, anal squamous cancer, and mesothelioma
  • Arm 3: Histological or blood-based confirmation of KRAS G12C mutation
Not Eligible

You will not qualify if you...

  • Has not recovered to CTCAE Grade 1 or better from adverse events due to cancer treatments administered more than 4 weeks earlier
  • History of a second malignancy unless treated with no evidence of disease for 2 years
  • History of hyperparathyroidism or hypercalcemia
  • Ophthalmological conditions including intraocular pressure >21 mm Hg or diagnosis of glaucoma, central serous retinopathy, retinal vein or artery occlusion, or retinal degenerative disease
  • Clinically significant cardiovascular disease
  • Bullous exfoliative skin disorders of any grade
  • Known hypersensitivity to MK-0472, MK-1084, pembrolizumab, or their ingredients
  • Use of proton-pump inhibitors or H2 histamine blockers within 7 days before first study dose
  • Discontinued prior anti-PD-1, anti-PD-L1, or related therapies due to adverse events
  • Received systemic anticancer therapy or investigational agents within 4 weeks before first dose
  • Received live or live-attenuated vaccines within 30 days before first dose
  • Used investigational agents or devices within 4 weeks before study treatment
  • Diagnosis of immunodeficiency or use of systemic steroids or immunosuppressive therapy within 7 days before first dose
  • Known progressing additional malignancy requiring treatment within past 2 years
  • Active central nervous system metastases or carcinomatous meningitis, unless stable for at least 4 weeks without steroids
  • Active autoimmune disease requiring systemic treatment in past 2 years except replacement therapy
  • History or current pneumonitis/interstitial lung disease requiring steroids
  • Active infection needing systemic therapy
  • History of allogeneic tissue or solid organ transplant
  • Not recovered from major surgery or ongoing surgical complications

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 25 locations

1

Northwestern Memorial Hospital ( Site 0002)

Chicago, Illinois, United States, 60611

Actively Recruiting

2

The University of Louisville, James Graham Brown Cancer Center ( Site 0004)

Louisville, Kentucky, United States, 40202

Actively Recruiting

3

John Theurer Cancer Center at Hackensack University Medical Center ( Site 0001)

Hackensack, New Jersey, United States, 07601

Actively Recruiting

4

Rutgers Cancer Institute of New Jersey ( Site 0005)

New Brunswick, New Jersey, United States, 08901

Actively Recruiting

5

Princess Margaret Cancer Centre ( Site 0101)

Toronto, Ontario, Canada, M5G 2M9

Actively Recruiting

6

Centre Hospitalier de l'Université de Montréal-Unit for Innovative Therapies ( Site 0100)

Montreal, Quebec, Canada, H2X 0A9

Actively Recruiting

7

Jewish General Hospital ( Site 0104)

Montreal, Quebec, Canada, H3T 1E2

Actively Recruiting

8

Centro de Estudios Clínicos SAGA ( Site 0701)

Santiago, Region M. de Santiago, Chile, 7500653

Actively Recruiting

9

Fundacion Arturo Lopez Perez ( Site 0700)

Santiago, Region M. de Santiago, Chile, 7500921

Actively Recruiting

10

Centro de Investigacion Clinicadela Universidad Catolica ( Site 0703)

Santiago, Region M. de Santiago, Chile, 8330034

Actively Recruiting

11

Bradfordhill ( Site 0702)

Santiago, Region M. de Santiago, Chile, 8420383

Actively Recruiting

12

Rambam Health Care Campus ( Site 0304)

Haifa, Israel, 3109601

Actively Recruiting

13

Shaare Zedek Medical Center ( Site 0303)

Jerusalem, Israel, 9103102

Actively Recruiting

14

Rabin Medical Center ( Site 0301)

Petah Tikva, Israel, 4941492

Actively Recruiting

15

Sheba Medical Center ( Site 0300)

Ramat Gan, Israel, 5265601

Actively Recruiting

16

Sourasky Medical Center ( Site 0302)

Tel Aviv, Israel, 6423906

Actively Recruiting

17

Narodowy Instytut Onkologii im. Marii Sklodowskiej-Curie - Panstwowy Instytut Badawczy w Warszawie ( Site 0401)

Warsaw, Masovian Voivodeship, Poland, 02-781

Actively Recruiting

18

Uniwersyteckie Centrum Kliniczne ( Site 0400)

Gdansk, Pomeranian Voivodeship, Poland, 80-214

Actively Recruiting

19

Institut Català d'Oncologia - L'Hospitalet-Medical Oncology ( Site 0501)

L'Hospitalet de Llobregat, Catalonia, Spain, 08907

Actively Recruiting

20

Centro Integral Oncologico Clara Campal-Hospital HM Universitario Sanchinarro-START Madrid, ( Site 0504)

Madrid, Madrid, Comunidad de, Spain, 28050

Actively Recruiting

21

Hospital Universitari Vall d'Hebron ( Site 0500)

Barcelona, Spain, 08035

Actively Recruiting

22

Hospital Virgen del Rocio ( Site 0503)

Seville, Spain, 41013

Actively Recruiting

23

Hôpitaux Universitaires de Genève (HUG) ( Site 0202)

Geneva, Canton of Geneva, Switzerland, 1211

Actively Recruiting

24

Cantonal Hospital St.Gallen-Oncology & Hematology ( Site 0201)

Sankt Gallen, Canton of St. Gallen, Switzerland, 9000

Actively Recruiting

25

Ospedale Regionale Bellinzona e Valli ( Site 0200)

Bellinzona, Canton Ticino, Switzerland, 6500

Actively Recruiting

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Research Team

T

Toll Free Number

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

3

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