Actively Recruiting

Phase 1
Phase 2
Age: 18Years +
All Genders
NCT04683250

Study of RET Inhibitor TAS0953/HM06 in Patients With Advanced Solid Tumors With RET Gene Abnormalities

Led by Taiho Pharmaceutical Co., Ltd. · Updated on 2026-03-03

244

Participants Needed

21

Research Sites

532 weeks

Total Duration

On this page

Sponsors

T

Taiho Pharmaceutical Co., Ltd.

Lead Sponsor

L

Linical Co., Ltd.

Collaborating Sponsor

AI-Summary

What this Trial Is About

Phase 1 and 2 trial to study the safety, pharmacokinetics, and efficacy of TAS0953/HM06 in patients with advanced solid tumors with RET gene abnormalities. Phase 1 aims to determine the Maximum Tolerated Dose (MTD) and identify the Recommended Phase 2 Dose (RP2D) to be used in phase 2.

CONDITIONS

Official Title

Study of RET Inhibitor TAS0953/HM06 in Patients With Advanced Solid Tumors With RET Gene Abnormalities

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Adult patient as defined by regional regulatory requirements
  • Eastern Cooperative Oncology Group (ECOG) performance score of 0 to 2
  • Presence of RET gene abnormalities confirmed by tissue or liquid biopsy
  • Adequate blood, liver, and kidney function
  • Advanced solid tumors for Phase 1 dose-escalation, with measurable or non-measurable disease
  • Asymptomatic brain or leptomeningeal metastases if present
  • For Phase 1 dose-expansion NSCLC patients with RET gene fusion: Cohorts 1 and 3 must be naive to RET inhibitors and no prior systemic anti-cancer treatment (except completed neo-adjuvant or adjuvant chemotherapy at least 6 months before)
  • For Phase 1 dose-expansion NSCLC patients with RET gene fusion: Cohorts 2 and 4 may have prior RET inhibitor exposure
  • Measurable disease per RECIST 1.1
  • For Phase 2: locally advanced or metastatic NSCLC patients with or without prior RET inhibitor exposure, or advanced solid tumors with RET abnormalities who have exhausted other treatments
Not Eligible

You will not qualify if you...

  • Use of investigational or anticancer therapy within 5 half-lives before starting study drug
  • Major surgery (except vascular access placement) within 4 weeks before starting study drug or planned during study
  • Whole brain radiotherapy within 14 days or other palliative radiotherapy within 7 days before starting study drug, or ongoing side effects from such therapy
  • Uncontrolled or significant cardiovascular diseases including recent heart attack, unstable angina, severe heart failure, or severe uncontrolled hypertension
  • QT interval corrected with Fridericia's formula >470 msec, history or risk factors for prolonged QT syndrome or Torsades de pointes
  • Treatment with strong CYP3A4 inhibitors within 1 week or inducers within 3 weeks before study drug start
  • Presence of known activating mutations in EGFR, KRAS, ALK, HER2, ROS1, BRAF, or METex14 (Phase 1 dose-expansion and Phase 2)

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 21 locations

1

Chao Family Comprehensive Cancer Center

Orange, California, United States, 92868-3298

Terminated

2

Stanford Cancer Center

Stanford, California, United States, 94305-5826

Terminated

3

Massachusetts General Hospital

Boston, Massachusetts, United States, 02114

Terminated

4

Henry Ford Hospital

Detroit, Michigan, United States, 48202

Terminated

5

START Midwest - Cancer & Hematology Centers of Western Michigan

Grand Rapids, Michigan, United States, 49546

Terminated

6

Laura and Isaac Perlmutter Cancer Center at NYU Langone Health

New York, New York, United States, 10016

Terminated

7

Memorial Sloan Kettering Cancer Center

New York, New York, United States, 10065

Terminated

8

The Sarah Cannon Research Institute/Tennessee Oncology

Nashville, Tennessee, United States, 37203

Terminated

9

The University of Texas M. D. Anderson Cancer Center

Houston, Texas, United States, 77030-4009

Terminated

10

National Cancer Center Hospital East

Kashiwa-shi, Chiba, Japan

Actively Recruiting

11

Tohoku University Hospital

Sendai, Miyagi, Japan

Actively Recruiting

12

Okayama University Hospital

Okayama, Okayama-ken, Japan

Actively Recruiting

13

Kansai Medical University Hospital

Hirakata-shi, Osaka, Japan

Actively Recruiting

14

Osaka International Cancer Institute

Osaka, Osaka, Japan

Actively Recruiting

15

Shizuoka Cancer Center

Shizuoka, Shizuoka, Japan

Actively Recruiting

16

National Cancer Center Hospital

Chuo-ku, Tokyo, Japan, 104-0045

Actively Recruiting

17

The Cancer Institute Hospital of JFCR

Koto-ku, Tokyo, Japan, 135-8550

Actively Recruiting

18

National Hospital Organization Kyushu Cancer Center

Fukuoka, Japan

Actively Recruiting

19

Kanagawa Cancer Center

Kanagawa, Japan

Actively Recruiting

20

Kurashiki Central Hospital

Okayama, Japan

Actively Recruiting

21

Samsung Medical Center

Seoul, South Korea

Actively Recruiting

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Research Team

K

Kazuo Koba

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SEQUENTIAL

Primary Purpose

TREATMENT

Number of Arms

2

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Study of RET Inhibitor TAS0953/HM06 in Patients With Advanced Solid Tumors With RET Gene Abnormalities | DecenTrialz