Actively Recruiting

Phase 2
Age: 18Years - 75Years
All Genders
NCT06029972

Study of Tilpisertib Fosmecarbil in Participants With Moderately to Severely Active Ulcerative Colitis

Led by Gilead Sciences · Updated on 2026-02-11

176

Participants Needed

129

Research Sites

217 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

The goal of this study is to learn if tilpisertib fosmecarbil (formerly known as GS-5290) is effective and safe in treating participants with moderate to severe ulcerative colitis. The study will compare participants in different treatment groups treated with tilpisertib fosmecarbil with participants treated with placebo. The primary objective of this study is to demonstrate the efficacy of tilpisertib fosmecarbil, compared to placebo control, in achieving Clinical Response at Week 12.

CONDITIONS

Official Title

Study of Tilpisertib Fosmecarbil in Participants With Moderately to Severely Active Ulcerative Colitis

Who Can Participate

Age: 18Years - 75Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Individuals assigned male at birth, or nonpregnant, nonlactating individuals assigned female at birth, aged 18 to 75 years
  • Ulcerative colitis diagnosed for at least 90 days before randomization, confirmed by endoscopy and histology
  • Disease extent of at least 15 cm from the anal verge
  • Moderately to severely active ulcerative colitis with a modified Mayo Clinic Score of 5 to 9 and an endoscopic subscore of 2 to 3
  • Previous treatment with at least one advanced therapy mechanism for ulcerative colitis but failure of no more than 3 different advanced therapies
  • Surveillance colonoscopy for dysplasia if indicated by regional guidelines prior to randomization
Not Eligible

You will not qualify if you...

  • Current diagnosis of Crohn's Disease, indeterminate colitis, lymphocytic or collagenous colitis
  • Disease limited to the rectum (ulcerative proctitis) at screening endoscopy
  • Ongoing therapy with or prior use of any prohibited medications
  • Active clinically significant infection, or infection requiring hospitalization or intravenous anti-infectives within 8 weeks
  • Infection requiring oral anti-infective therapy within 6 weeks of randomization
  • History of opportunistic infection
  • Current diagnosis of acute severe colitis, fulminant colitis, or toxic megacolon

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 129 locations

1

GI Alliance

Sun City, Arizona, United States, 85351

Actively Recruiting

2

GastroSb Weight Loss Clinic

Chula Vista, California, United States, 91910

Actively Recruiting

3

Southern California Research Centers

Coronado, California, United States, 92118

Actively Recruiting

4

VVCRD Research

Garden Grove, California, United States, 92845

Actively Recruiting

5

UC San Diego Health System

La Jolla, California, United States, 92037

Actively Recruiting

6

Gastro Care Institute

Lancaster, California, United States, 93534

Actively Recruiting

7

Om Research LLC

Lancaster, California, United States, 93534

Actively Recruiting

8

United Medical Doctors

Murrieta, California, United States, 92563

Withdrawn

9

University of California, Davis

Sacramento, California, United States, 95817

Actively Recruiting

10

University of California San Francisco

San Francisco, California, United States, 94115

Actively Recruiting

11

Amicis Research Center

Valencia, California, United States, 91355

Withdrawn

12

Luna Research

Coral Gables, Florida, United States, 33134

Actively Recruiting

13

University of Florida

Gainesville, Florida, United States, 32610

Actively Recruiting

14

The Medici Medical Research

Hollywood, Florida, United States, 33021

Actively Recruiting

15

Encore Medical Research, LLC

Hollywood, Florida, United States, 33024

Withdrawn

16

Clinical Research of Osceola

Kissimmee, Florida, United States, 34741

Actively Recruiting

17

Florida Research Institute

Largo, Florida, United States, 33771

Actively Recruiting

18

Wellness Research Center

Miami, Florida, United States, 33135

Withdrawn

19

IMIC Inc

Miami, Florida, United States, 33176

Withdrawn

20

Reserka LLC

Miami, Florida, United States, 33176

Withdrawn

21

GI PROS Research

Naples, Florida, United States, 34102

Actively Recruiting

22

Clinical One Research

Orlando, Florida, United States, 32807

Actively Recruiting

23

Digestive and Liver Center of Florida, LLC

Orlando, Florida, United States, 32825

Actively Recruiting

24

Advanced Medical Research Center

Port Orange, Florida, United States, 32127

Actively Recruiting

25

Gastroenterology Associates of Florida - GI Alliance

Wellington, Florida, United States, 33414

Withdrawn

26

Atlanta Center For Gastroenterology P.C.

Decatur, Georgia, United States, 30033

Withdrawn

27

Corewell Health

Grand Rapids, Michigan, United States, 49546

Actively Recruiting

28

Mayo Clinic

Rochester, Minnesota, United States, 55905

Actively Recruiting

29

Gastroenterology Associates of North Mississippi

Oxford, Mississippi, United States, 38655

Actively Recruiting

30

Digestive Health Specialists

Tupelo, Mississippi, United States, 38801

Actively Recruiting

31

St. Charles Clinical Research

St Louis, Missouri, United States, 63141

Actively Recruiting

32

Ellipsis Research Group

Brooklyn, New York, United States, 11215

Active, Not Recruiting

33

NYU Langone Long Island Clinical Research Associates

Great Neck, New York, United States, 11021

Actively Recruiting

34

Gastroenterology & Hepatology Specialists Inc

Canton, Ohio, United States, 44718

Actively Recruiting

35

Ohio Gastroenterology & Liver Institute

Cincinnati, Ohio, United States, 45249

Withdrawn

36

The Ohio State University Wexner Medical Centre

Columbus, Ohio, United States, 43210

Actively Recruiting

37

Dayton Gastroenterology, LLC

Dayton, Ohio, United States, 45145

Actively Recruiting

38

Great Lakes Gastroenterology Research, LLC

Mentor, Ohio, United States, 44060

Actively Recruiting

39

Hightower Clinical

Oklahoma City, Oklahoma, United States, 73134

Withdrawn

40

Skyline Gastroenterology of West Tennessee

Jackson, Tennessee, United States, 38301

Not Yet Recruiting

41

Gastroenterology Research of Hill Country

Boerne, Texas, United States, 78006

Actively Recruiting

42

Gastroenterology Research of America

El Paso, Texas, United States, 79936

Withdrawn

43

DHAT Research Institute

Garland, Texas, United States, 75044

Withdrawn

44

Southwest Clinical Trials

Houston, Texas, United States, 77074

Withdrawn

45

GI Alliance

Lubbock, Texas, United States, 79410

Actively Recruiting

46

GI Associates and Endoscopy Center - GI Alliance

Mansfield, Texas, United States, 76063

Actively Recruiting

47

Clinical Associates in Research Therapeutics of America

San Antonio, Texas, United States, 78212

Actively Recruiting

48

Gastroenterology Research of San Antonio

San Antonio, Texas, United States, 78229

Actively Recruiting

49

Tyler Research Institute, LLC

Tyler, Texas, United States, 75701

Actively Recruiting

50

Gastroenterology Associates of Tidewater

Chesapeake, Virginia, United States, 23320

Actively Recruiting

51

Emeritas Group Research

Lansdowne Town Center, Virginia, United States, 20176

Actively Recruiting

52

Gastroenterology Consultants of Southwest Virginia

Roanoke, Virginia, United States, 24014

Actively Recruiting

53

Swedish Medical Center

Seattle, Washington, United States, 98122

Withdrawn

54

Sunshine Coast University Hospital

Birtinya, Queensland, Australia, 4575

Actively Recruiting

55

Mater Adult Hospital

South Brisbane, Queensland, Australia, 4101

Actively Recruiting

56

Princess Alexandra Hospital

Woolloongabba, Queensland, Australia, 4102

Actively Recruiting

57

Royal Adelaide Hospital

Adelaide, South Australia, Australia, 5000

Actively Recruiting

58

Queen Elizabeth Hospital

Woodville, South Australia, Australia, 5011

Actively Recruiting

59

Monash Medical Centre

Clayton, Victoria, Australia, 3168

Withdrawn

60

Northern Health

Epping, Victoria, Australia, 3076

Actively Recruiting

61

Footscray Hospital

Footscray, Victoria, Australia, 3011

Actively Recruiting

62

Fiona Stanley Hospital

Murdoch, Western Australia, Australia, 6150

Actively Recruiting

63

Medical University of Innsbruck

Innsbruck, Austria, 6020

Actively Recruiting

64

University of Salzburg, Universitätsklinik für Innere Medizin III

Salzburg, Austria, 5020

Not Yet Recruiting

65

Universitätsklinikum St. Pölten

Sankt Pölten, Austria, 3100

Actively Recruiting

66

Medical University Vienna, Department of Internal Medicine III, Division Gastroenterology and Hepatology

Vienna, Austria, 1090

Actively Recruiting

67

Universitaire Ziekenhuis Leuven

Leuven, Belgium, 3000

Actively Recruiting

68

London Health Sciences Centre-University Hospital

London, Canada, N6A 5A5

Actively Recruiting

69

Physician's Clinical Research, Inc. (PCRI)

Toronto, Canada, M2K 2W2

Withdrawn

70

Mount Sinai Hospital

Toronto, Canada, MSG 1X5

Actively Recruiting

71

TDDA Speciality Research

Vaughan, Canada, L4L 4Y7

Actively Recruiting

72

Centre Hospitalier Universitaire Grenoble

Grenoble, France, 38043

Actively Recruiting

73

Hôpital Claude Huriez

Little Cedex, France, 59037

Actively Recruiting

74

Hopital Saint Eloi

Montpellier, France, 34295

Actively Recruiting

75

Centre Hospitalier Universitaire de Nantes

Nantes, France, 44000

Actively Recruiting

76

Institut des MICI

Neuilly-sur-Seine, France, 92200

Actively Recruiting

77

CHU de Saint Etienne - Hopital Nord

Saint-Etienne, France, 42055

Actively Recruiting

78

Hopital Rangueil

Toulouse, France, 31059

Actively Recruiting

79

CHRU Nancy

Vandœuvre-lès-Nancy, France, 54500

Actively Recruiting

80

Charite Universitaetsmedizin Berlin Campus CVK, Department of Hepatology and Gastroenterology

Berlin, Germany, 13353

Not Yet Recruiting

81

Medizinische Hochschule Hannover

Hanover, Germany, 30625

Not Yet Recruiting

82

Universitatsklinikum Schleswig-Holstein

Kiel, Germany, 24105

Actively Recruiting

83

Eugastro Gmbh

Liepzig, Germany, 4103

Actively Recruiting

84

Universitaetsklinikum Ulm Klinik fur Innere Medizin I CED Studien Ambulanz

Ulm, Germany, 89081

Not Yet Recruiting

85

Tolna Megye Balassa Janos Korhaz

Beri Balogh, Hungary, 7100

Actively Recruiting

86

Szent Janos Korhaz es Eszak-budai Egyesitett Korhazak

Budapest, Hungary, 1033

Actively Recruiting

87

AZIENDA UNICA OSPEDALIERO-UNIVERSITARIA"RENATO DULBECCO" - AOU"Mater Domini"

Catanzaro, Italy, 88100

Actively Recruiting

88

IRCCS Istituto Clinico Humanitas

Milan, Italy, 20089

Actively Recruiting

89

Azienda Ospedaliera San Camillo Forlanini

Roma, Italy, 00152

Actively Recruiting

90

Istituto Clinico Humanitas

Rozzano, Italy, 20089

Actively Recruiting

91

Azienda Sanitaria Universitaria Friuli Centrale

Udine, Italy, 33100

Withdrawn

92

Hyogo Medical University Hospital

Hyōgo, Japan, 663-8501

Actively Recruiting

93

Fukuoka University Hospital

Jonan-ku, Japan, 814-0180

Actively Recruiting

94

The Jikei University Hospital

Minatoku, Japan, 105-8471

Actively Recruiting

95

Kitasato University Kitasato Institute Hospital

Minatoku, Japan, 108-8642

Actively Recruiting

96

Kyorin University Hospital

Mitaka-shi, Japan, 181-8611

Actively Recruiting

97

Nagasaki University Hospital

Nagasaki, Japan, 852-8501

Actively Recruiting

98

Ishida Clinic of IBD and Gastroenterology

Ōita, Japan, 870-0823

Actively Recruiting

99

Saga University Hospital

Sagaken, Japan, 849-8501

Actively Recruiting

100

Kitasato University Hospital

Sagamihara, Japan, 252-0375

Actively Recruiting

101

Sapporo Medical University Hospital

Sapporo, Japan, 060-8543

Actively Recruiting

102

Ginza Central Clinic

Tokyo, Japan, 104-0061

Actively Recruiting

103

Institute of Science Tokyo Hospital

Toukiyouto, Japan, 113-8519

Actively Recruiting

104

Economicus Sp. z o.o., Niepubliczny Zakład Opieki Zdrowotnej (NZOZ) ALL-MEDICUS

Katowice, Poland, 40-659

Withdrawn

105

Gabinet Endoskopii Przewodu Pokarmowego

Krakow, Poland, 31-009

Actively Recruiting

106

Medrise Sp. z o.o. Centrum Badań Klinicznych

Lublin, Poland, 20-852

Not Yet Recruiting

107

SOLUMED Centrum Medyczne

Poznan, Poland, 60-425

Not Yet Recruiting

108

Kliniczny Szpital Wojewódzki Nr 2 im. Sw. Jadwigi Królowej w Rzeszowie

Rzeszów, Poland, 35-210

Actively Recruiting

109

Specjalistyczna Praktyka Lekarska Leszek Bryniarski

Sopot, Poland, 81-756

Actively Recruiting

110

GASTROMED Kopon, Zmudzinski i wspolnicy Sp. J. Specialized Center of Gastroenterology and Endoscopy

Torun, Poland, 87-100

Actively Recruiting

111

Medical Network Sp. z o.o. WIP Warsaw IBD Point Profesor Kierkus

Warsaw, Poland, 00-728

Actively Recruiting

112

Nzoz Vivamed

Warsaw, Poland, 03-580

Withdrawn

113

Specjalistyczne Gabinety Lekarskie Body Clinic

Warsaw, Poland, 03-712

Actively Recruiting

114

Centrum Medyczne Oporow

Wroclaw, Poland, 52-416

Actively Recruiting

115

Yonsei University Severance Hospital

Seodaemun-Gu, VIC, South Korea, 3772

Actively Recruiting

116

Inje University

Busan, South Korea, 48108

Actively Recruiting

117

Yeungnam University Hospital

Daegu, South Korea, 42415

Actively Recruiting

118

Kyungpook National University Hospital

Junggu, South Korea, 41944

Actively Recruiting

119

Kyung Hee University Medical Center

Seoul, South Korea, 02447

Actively Recruiting

120

Kangbuk Samsung Hospital

Seoul, South Korea, 03181

Actively Recruiting

121

Hanyang University Hospital

Seoul, South Korea, 04763

Actively Recruiting

122

Samsung Medical Center

Seoul, South Korea, 06351

Actively Recruiting

123

Wonju Severance Christian Hospital

Wŏnju, South Korea, 26426

Actively Recruiting

124

Intesto, Gastroenterologische Praxis Crohn-Colitis-Zentrum

Bern, Switzerland, 3012

Actively Recruiting

125

Fairfield General Hospital

Bury, United Kingdom, BL9 7TD

Actively Recruiting

126

Cambridge University Hospitals NHS Foundation Trust

Cambridge, United Kingdom, CB2 0QQ

Actively Recruiting

127

Barts Health NHS Trust

London, United Kingdom, E1 2AJ

Actively Recruiting

128

Norfolk and Norwich University Hospital Nhs Foundation Trust

Norwich, United Kingdom, NR4 7UZ

Actively Recruiting

129

University Hospital Southampton Nhs Foundation Trust

Southampton, United Kingdom, SO16 6YD

Actively Recruiting

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Research Team

G

Gilead Clinical Study Information Center

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

DOUBLE

Allocation

RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

4

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