Actively Recruiting

Phase 1
Age: 18Years +
MALE
NCT07244341

A Study of Valemetostat (DS-3201b) in Combination With Darolutamide in Metastatic Castration Resistant Prostate Cancer (mCRPC)

Led by Daiichi Sankyo · Updated on 2026-02-04

60

Participants Needed

6

Research Sites

208 weeks

Total Duration

On this page

Sponsors

D

Daiichi Sankyo

Lead Sponsor

B

Bayer

Collaborating Sponsor

AI-Summary

What this Trial Is About

This study will assess the safety and tolerability of valemetostat in combination with darolutamide in participants with Metastatic Castration Resistant Prostate Cancer (mCRPC).

CONDITIONS

Official Title

A Study of Valemetostat (DS-3201b) in Combination With Darolutamide in Metastatic Castration Resistant Prostate Cancer (mCRPC)

Who Can Participate

Age: 18Years +
MALE

Eligibility Criteria

Eligible

You may qualify if you...

  • Adult males 18 years of age or older at the time of consent
  • Histologically confirmed adenocarcinoma of the prostate including neuroendocrine differentiation except pure small cell carcinoma
  • Evidence of disease progression per PCWG3 modified RECIST v1.1 criteria
  • Radiographic confirmation of metastatic disease by CT, MRI, or bone scan
  • Ongoing androgen deprivation therapy initiated at least 4 weeks prior and continued during the trial
  • Baseline PSA level of 2 ng/mL or higher
  • Prior therapy with androgen receptor pathway inhibitors
  • ECOG performance status of 0 or 1 within 28 days prior to enrollment
  • Willing and able to provide adequate fresh or archival tumor samples; pretreatment biopsy required if not contraindicated
  • If capable of producing sperm, agrees to use contraception and not donate or freeze sperm during and for 3 months after treatment
Not Eligible

You will not qualify if you...

  • Prior treatment with epigenetic agents including EZH1, EZH2, EZH1/2, or PRC2 inhibitors
  • Presence of super scan on baseline bone scan
  • Clinically active brain metastases, spinal cord compression, or leptomeningeal carcinomatosis requiring treatment
  • Uncontrolled or significant cardiovascular disease
  • Prior malignancy active within the past 3 years except certain locally curable cancers
  • Active or uncontrolled hepatitis B infection
  • Active or uncontrolled hepatitis C infection
  • Active or uncontrolled HIV infection

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Trial Site Locations

Total: 6 locations

1

Carolina Urologic Research Center

Myrtle Beach, South Carolina, United States, 29572-4607

Actively Recruiting

2

NEXT Oncology

San Antonio, Texas, United States, 78229-6028

Actively Recruiting

3

Virginia Cancer Specialists (NEXT Virginia)

Fairfax, Virginia, United States, 22031-2171

Actively Recruiting

4

Kobe City Med Cen Gen Hosp.

Kobe, Japan, 650-0047

Actively Recruiting

5

Cancer Institute Hospital of JFCR

Kōtoku, Japan, 135-8550

Actively Recruiting

6

Toho University Sakura Medical Center

Sakura-shi, Japan, 285-8741

Actively Recruiting

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Research Team

C

Contact for Trial Information

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NON_RANDOMIZED

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

2

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A Study of Valemetostat (DS-3201b) in Combination With Darolutamide in Metastatic Castration Resistant Prostate Cancer (mCRPC) | DecenTrialz