Actively Recruiting

Phase 1
Age: 18Years - 75Years
All Genders
NCT05772455

A Study of XZB-0004 in Patients With Solid Tumors

Led by Xuanzhu Biopharmaceutical Co., Ltd. · Updated on 2024-10-28

128

Participants Needed

1

Research Sites

201 weeks

Total Duration

On this page

AI-Summary

What this Trial Is About

XZB-0004 is a novel and potent small molecule inhibitor of receptor tyrosine kinase AXL. This is an open-label, multicentre phase I study of XZB-0004 in patients with solid tumors. Part 1 is a dose-escalation study to evaluate the safety, pharmacokinetic (PK), and pharmacodynamic profile of XZB-0004, and then to identify a safe and pharmacologically active dose for evaluation in subsequent cohorts or clinical studies. Part 2 is a study to evaluate the efficacy and safety of XZB-0004 combined with Penpulimab in patients with NSCLC or advanced solid tumors.

CONDITIONS

Official Title

A Study of XZB-0004 in Patients With Solid Tumors

Who Can Participate

Age: 18Years - 75Years
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Patient has signed informed consent before any trial related activities.
  • Be 18 years of age or older and less than 75 years at the time of signing the informed consent.
  • Part 1: Have a histologically or cytologically confirmed diagnosis of a solid tumour malignancy; Part 2: Have a histologically or cytologically confirmed diagnosis of NSCLC or solid tumour malignancy.
  • Have evaluable (for Part 1) or measurable (for Part 2) disease as the Response Evaluation Criteria in Solid Tumours (RECIST) 1.1.
  • Have a performance status score of 0 or 1 according to the Eastern Cooperative Oncology Group (ECOG) scale.
  • Have adequate organ function.
  • Have recovered to 64 grade 1 or meet the study requirements from effects of prior cancer therapy, except alopecia; irreversible neuropathy should have recovered to 64 grade 2.
  • Have a life expectancy greater than 3 months.
  • Eligible patients who are fertile must agree to use a reliable contraceptive method with their partner.
  • Willingness to comply with scheduled visits, treatment plans, laboratory tests, and other study procedures.
Not Eligible

You will not qualify if you...

  • Previous use of AXL inhibitors and immunotherapy inconsistent with protocol requirements.
  • Received anti-tumor therapy such as chemotherapy, radiotherapy, biotherapy, endocrine therapy, immunotherapy, or other therapy within 4 weeks prior to the first dose.
  • Received unmarketed investigational drugs or treatments within 4 weeks or 5 times the elimination half-life before the first dose.
  • Treatment with systemic glucocorticoids (prednisone > 10mg per day or equivalent) or other immunosuppressive agents within 14 days before the first dose.
  • Inability to swallow, intestinal obstruction, or other factors affecting drug absorption.
  • Patient with impaired heart function or clinically significant heart disease.
  • Any condition or illness that would interfere with safety evaluation.
  • History of immune deficiencies, including positive HIV antibody tests.
  • Patient is in the active stage of HBV or HCV.
  • History of solid organ or bone marrow transplant.
  • Any other malignant tumor diagnosed within 5 years.
  • Known primary tumor of the central nervous system or CNS metastases.
  • Uncontrolled pleural effusion, pericardial effusion, or ascites requiring repeated drainage within 4 weeks before dosing.
  • Psychiatric disorders that may affect trial compliance.
  • History of alcoholism or drug abuse.
  • Pregnant or breastfeeding.
  • Cases deemed unsuitable for inclusion by researchers.

AI-Screening

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Trial Site Locations

Total: 1 location

1

Shanghai Pulmonary Hospital

Shanghai, Shanghai Municipality, China, 200433

Actively Recruiting

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Research Team

X

Xiujie Zhang

CONTACT

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

NA

Model

SINGLE_GROUP

Primary Purpose

TREATMENT

Number of Arms

1

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