Actively Recruiting

Early Phase 1
Age: 18Years +
All Genders
ID05804227

Window-of-Opportunity Trial of Ulixertinib for MAPK-Activated Gliomas

Led by M.D. Anderson Cancer Center · Updated on 2026-02-27

40

Participants Needed

1

Research Sites

N/A

Total Duration

On this page

Sponsors

M

M.D. Anderson Cancer Center

Lead Sponsor

B

BioMed Valley Discoveries, Inc

Collaborating Sponsor

AI-Summary

What this Trial Is About

Researchers are investigating the ability of the drug ulixertinib to cross the blood-brain barrier in patients with recurrent MAPK-activated gliomas, a type of brain tumor. The study aims to evaluate how well ulixertinib penetrates the tumor and cerebrospinal fluid, and to assess its anti-tumor activity, safety, and tolerability. This early-phase trial is sponsored by M.D. Anderson Cancer Center and involves patients with specific genetic mutations in their gliomas. Participants are divided into two groups: surgical and non-surgical. Adults in the surgical group will take ulixertinib by mouth twice daily for two weeks before undergoing tumor removal surgery around day 14. The non-surgical group, which includes patients aged 12 and older, will take ulixertinib orally twice daily continuously in 28-day treatment cycles. Pediatric dosing is adjusted based on body surface area. During the study, participants will undergo evaluations including tumor and plasma drug concentration measurements, imaging to assess disease progression, and monitoring for side effects using established criteria. Researchers will also track progression-free survival, overall survival, response duration, and time to next treatment. The study includes safety assessments throughout and plans to monitor patients for an average of one year after starting treatment.

CONDITIONS

Brief Title

Window-of-Opportunity Trial of Ulixertinib for MAPK-Activated Gliomas

Who Can Participate

Age: 18Years +
All Genders

Eligibility Criteria

Eligible

You may qualify if you...

  • Willing and able to provide written informed consent or assent, with legally authorized representative consent if cognitively impaired
  • Surgical group: 18 years or older; Non-surgical group: 12 years or older
  • Pediatric patients must have body surface area of at least 0.9 m2 for accurate dosing
  • Diagnosis of MAPK-activated gliomas or related tumors confirmed by pathology or genetic testing
  • Prior tumor resection or biopsy confirming glioma diagnosis
  • Low grade gliomas must have prior radiation or chemotherapy; high grade gliomas must have prior radiation
  • Progressive disease per imaging criteria and presence of resectable tumor for surgical group
  • At least 12 weeks from radiation with evidence of disease progression
  • Any number of prior relapses
  • Willing to provide archival tissue samples
  • Performance status of 60 or higher on the Karnofsky Performance Scale
  • Stable or decreasing steroid dose, not exceeding 16mg dexamethasone or equivalent daily
  • Adequate organ function per specified laboratory values
  • Negative pregnancy test for females of childbearing potential
  • Agreement to use effective contraception during the study and for 90 days after last treatment
Not Eligible

You will not qualify if you...

  • Treatment with bevacizumab within 3 months prior to enrollment
  • Presence of implanted chemotherapy (unless previously resected)
  • Less than 12 weeks since completing radiotherapy without biopsy-proven progression
  • Participation in another investigational study or use of investigational devices
  • Severe immunodeficiency or recent systemic immunosuppressive therapy (except steroids)
  • Recent chemotherapy or targeted therapy within 3 weeks before study start without recovery
  • Additional active malignancies requiring treatment, except certain skin or cervical cancers
  • Active infections needing systemic therapy
  • Conditions or abnormalities interfering with trial participation or results
  • Psychiatric or substance abuse disorders affecting cooperation
  • Pregnancy, breastfeeding, or planning to conceive during the study
  • Contraindications for MRI procedures
  • Not eligible for non-emergent surgical resection
  • Use of prohibited medications unable to be discontinued prior to enrollment
  • History or risk of retinal vein occlusion or central serous retinopathy

AI-Screening

AI-Powered Screening

Complete this quick 3-step screening to check your eligibility

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Your Study Journey

Screening

Duration - 2 to 4 weeks

Participants are screened for eligibility to participate in the trial.

1 visit (in-person)

Treatment

Duration - Surgical: 2 weeks; Non-Surgical: cycles of 28 days ongoing

Participants in the surgical cohort take Ulixertinib by mouth twice daily for two weeks before undergoing tumor resection. Participants in the non-surgical cohort take Ulixertinib by mouth twice daily continuously in 28-day cycles.

Surgical: 1 baseline visit and 1 surgery visit; Non-Surgical: visits every 28 days per cycle

Trial Site Locations

Total: 1 location

1

M D Anderson Cancer Center

Houston, Texas, United States, 77030

Actively Recruiting

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Research Team

N

Nazanin Majd, MD

How is the study designed?

Study Type

INTERVENTIONAL

Masking

NONE

Allocation

RANDOMIZED

Model

PARALLEL

Primary Purpose

TREATMENT

Number of Arms

2

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